SCHEMBL5736843

SCHEMBL5736843

Cc1cccc(-c2nc(Nc3ccc4[nH]ncc4c3)c3ccc(Cl)cc3n2)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 9/20 0.56
TGFBR1 P36897 1/20 0.56
ROCK1 Q13464 2/20 0.52
PAK4 O96013 2/20 0.51
CLK2 P49760 1/20 0.51
BLK P51451 1/20 0.51
CSNK2A1 P68400 1/20 0.51
STK3 Q13188 1/20 0.51
DYRK1A Q13627 1/20 0.51
AURKB Q96GD4 1/20 0.51
CLK4 Q9HAZ1 1/20 0.51
STK17A Q9UEE5 1/20 0.51
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
AURKA O14965 1/20 0.50
GAA P10253 1/20 0.50
MAPT P10636 2/20 0.49
ABCG2 Q9UNQ0 2/20 0.49
ABCB1 P08183 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3581146 0.99 ROCK2 (0.56) ROCK2TGFBR1ROCK1PAK4CLK2
SCHEMBL3582617 0.92 ROCK2 (0.56) ROCK2TGFBR1ROCK1PAK4CLK2
SCHEMBL3581521 0.92 ROCK2 (0.58) ROCK2TGFBR1ROCK1PAK4CLK2
SCHEMBL3581577 0.89 TGFBR1 (0.54) ROCK2TGFBR1ROCK1PAK4CLK2
SCHEMBL3583464 0.89 ROCK2 (0.58) ROCK2TGFBR1ROCK1PAK4CLK2
SCHEMBL6925655 0.85 ROCK2 (0.54) ROCK2TGFBR1ROCK1PAK4CLK4
Trifluoroacetic Acid SCHEMBL3581419 0.84 ROCK2 (0.61) ROCK2TGFBR1ROCK1CLK2BLK
SCHEMBL3584500 0.83 PAK4 (0.51) ROCK2TGFBR1ROCK1PAK4CLK2
SCHEMBL18114600 0.83 ROCK2 (0.59) ROCK2TGFBR1ROCK1CLK2BLK
SCHEMBL13319629 0.83 MEN1 (0.60) ROCK2TGFBR1ROCK1CLK2BLK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1370553-B1 RHO-KINASE INHIBITORS BAYER AG (US) 2006-05-10 EP claimed