SCHEMBL6925655

SCHEMBL6925655

Clc1ccc2c(Nc3ccc4[nH]ncc4c3)nc(-c3cccnc3)nc2c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 4/20 0.54
PAK4 O96013 2/20 0.52
CYP1A2 P05177 2/20 0.51
CYP3A4 P08684 2/20 0.51
TSHR P16473 2/20 0.51
USP2 O75604 1/20 0.51
ALDH1A1 P00352 1/20 0.51
LMNA P02545 1/20 0.51
CLK4 Q9HAZ1 1/20 0.51
MAPT P10636 2/20 0.51
MAPK1 P28482 2/20 0.51
KDM4E B2RXH2 1/20 0.51
HPGD P15428 1/20 0.51
CYP2C19 P33261 1/20 0.51
HSD17B10 Q99714 1/20 0.51
TDP1 Q9NUW8 1/20 0.51
ABCG2 Q9UNQ0 7/20 0.50
TGFBR1 P36897 1/20 0.50
ABCB1 P08183 2/20 0.49
HTT P42858 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL3585583 0.91 ROCK2 (0.55) ROCK2PAK4CYP1A2CYP3A4TSHR
SCHEMBL3583464 0.90 ROCK2 (0.58) ROCK2PAK4CLK4KDM4EABCG2
SCHEMBL3581521 0.89 ROCK2 (0.58) ROCK2PAK4CLK4KDM4EABCG2
SCHEMBL6694965 0.88 MAPT (0.60) ROCK2CYP1A2CYP3A4TSHRUSP2
SCHEMBL5736843 0.85 ROCK2 (0.56) ROCK2PAK4CLK4MAPTABCG2
Hydrochloric Acid SCHEMBL3581146 0.85 ROCK2 (0.56) ROCK2PAK4CLK4MAPTABCG2
SCHEMBL3584500 0.84 PAK4 (0.51) ROCK2PAK4CLK4ABCG2TGFBR1
SCHEMBL3581577 0.84 TGFBR1 (0.54) ROCK2PAK4LMNACLK4MAPT
SCHEMBL14473992 0.83 CYP1A2 (0.57) CYP1A2CYP3A4TSHRUSP2ALDH1A1
SCHEMBL14474125 0.83 ABCG2 (0.65) CYP1A2CYP3A4TSHRUSP2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004065392-A1 CONDENSED PYRIDINES AND PYRIMIDINES AND THEIR USE AS ALK-5 RECEPTOR LIGANDS SMITHKLINE BEECHAM CORPORATION (US) 2004-08-05 WO disclosed