SCHEMBL5738889

SCHEMBL5738889

O=C(O)CCN(I)NS(=O)(=O)c1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TBXA2R P21731 2/20 0.50
ALDH1A1 P00352 2/20 0.50
MMP9 P14780 2/20 0.44
MMP8 P22894 2/20 0.44
MMP13 P45452 2/20 0.44
MMP1 P03956 2/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
MMP2 P08253 1/20 0.44
MAPT P10636 2/20 0.43
PTGES O14684 1/20 0.43
ADAMTS4 O75173 1/20 0.42
GAA P10253 2/20 0.41
MMP12 P39900 1/20 0.41
BCAT1 P54687 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
KDM4E B2RXH2 1/20 0.41
KAT6A Q92794 1/20 0.40
ATM Q13315 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1200801 0.72 ALDH1A1 (0.75) TBXA2RALDH1A1MMP9MMP13MMP2
SCHEMBL11796476 0.70 MAPK1 (0.53) TBXA2RALDH1A1MMP9MMP8MMP13
SCHEMBL16353991 0.70 EGFR (0.55) TBXA2RALDH1A1MMP9MMP8MMP13
Succinic Acid SCHEMBL19211914 0.69 TSHR (0.64) TBXA2RALDH1A1MMP9MMP8MMP13
SCHEMBL911198 0.69 ALDH1A1 (0.87) TBXA2RALDH1A1MAPTGAASMN1; SMN2
SCHEMBL11793418 0.69 MAPK1 (0.55) TBXA2RALDH1A1MMP9MMP8MMP13
SCHEMBL3864254 0.69 TBXA2R (0.45) TBXA2RALDH1A1
SCHEMBL3864255 0.69 ALDH1A1 (0.57) TBXA2RALDH1A1MMP9MMP8MMP13
Hydrazine SCHEMBL11854301 0.69 ALDH1A1 (0.71) TBXA2RALDH1A1MMP9MMP13MMP2
SCHEMBL5738891 0.69 ALDH1A1 (0.45) TBXA2RALDH1A1MAPTATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1331937-B1 DIBENZOXAZEPINE ALPHA V INTEGRIN RECEPTOR ANTAGONIST MERCK & CO INC (US) 2006-03-15 EP disclosed
EP-1044001-B1 INTEGRIN RECEPTOR ANTAGONISTS MERCK & CO INC (US) 2005-07-06 EP disclosed
CN-1284944-A Integrin receptor antagonists MERCK & CO INC (US) 2001-02-21 CN disclosed
CN-1284955-A Integrin receptor antagonists MERCK & CO INC (US) 2001-02-21 CN disclosed