SCHEMBL5740073

SCHEMBL5740073

COC(=O)C1Cc2ccccc2C(CCCS(=O)(=O)O)N1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 4/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
KDM4E B2RXH2 2/20 0.36
HSD17B10 Q99714 2/20 0.36
TSHR P16473 1/20 0.36
HTT P42858 1/20 0.36
OPRM1 P35372 3/20 0.33
CCKBR P32239 2/20 0.33
ALDH1A1 P00352 2/20 0.33
OPRK1 P41145 1/20 0.33
GRM7 Q14831 2/20 0.33
CYP1A2 P05177 1/20 0.33
GAA P10253 1/20 0.33
CYP2D6 P10635 1/20 0.33
MAPT P10636 1/20 0.33
CYP2C9 P11712 1/20 0.33
HPGD P15428 1/20 0.33
ALOX15 P16050 1/20 0.33
CYP2C19 P33261 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3249767 0.86 CYP2D6 (0.41) MEN1KMT2AKDM4ETSHROPRM1
SCHEMBL3240481 0.82 PDE5A (0.37) PDE5AMEN1KMT2AKDM4EHSD17B10
SCHEMBL7995094 0.71 ALDH1A1 (0.36) MEN1KMT2ATSHRALDH1A1CYP1A2
SCHEMBL917364 0.70 ALDH1A1 (0.52) KDM4EOPRM1ALDH1A1OPRK1GAA
SCHEMBL28209006 0.69 PDE5A (0.41) PDE5AMEN1KMT2AKDM4EHSD17B10
SCHEMBL28296124 0.68 GAA (0.35) MEN1KMT2ATSHROPRM1ALDH1A1
SCHEMBL918901 0.67 ALDH1A1 (0.51) KDM4EOPRM1ALDH1A1OPRK1GAA
SCHEMBL24177405 0.67 MEN1 (0.45) PDE5AMEN1KMT2AKDM4EHSD17B10
SCHEMBL4881527 0.67 PTPRA (0.36) MEN1KMT2AKDM4ETSHRHTT
SCHEMBL29365938 0.67 MEN1 (0.45) PDE5AMEN1KMT2AKDM4EHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1646659-B1 METHOD FOR THE PREPARATION OF 1,3-PROPANE DISULFONIC ACID COMPOUNDS KIACTA S RL (CH) 2014-05-14 EP disclosed
CN-101597196-A Improved drug candidate and preparation method thereof BELLUS HEALTH INTERNAT LTD (CH) 2009-12-09 CN disclosed
CN-100528840-C Improved drug candidates and methods for their preparation NEUROCHEM INTERNAT LTD (CH) 2009-08-19 CN disclosed
CN-1839117-A Improved drug candidates and methods for their preparation NEUROCHEM INTERNAT LTD (CH) 2006-09-27 CN disclosed
EP-1646659-A2 IMPROVED PHARMACEUTICAL DRUG CANDIDATES AND METHODS FOR PREPARATION THEREOF Neurochem (International) Limited (CH) 2006-04-19 EP disclosed
WO-2004113391-A2 IMPROVED PHARMACEUTICAL DRUG CANDIDATES AND METHODS FOR PREPARATION THEREOF NEUROCHEM (INTERNATIONAL) LIMITED (CH) 2004-12-29 WO disclosed