SCHEMBL28296124

SCHEMBL28296124

CCCC1NC(C(N)=O)Cc2ccccc21

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.35
MAPT P10636 1/20 0.35
PRCP P42785 1/20 0.35
MTNR1A P48039 2/20 0.34
MTNR1B P49286 2/20 0.34
TSHR P16473 2/20 0.34
MEN1 O00255 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
ALOX15 P16050 1/20 0.34
MAPK1 P28482 1/20 0.34
CYP2C19 P33261 1/20 0.34
KMT2A Q03164 1/20 0.34
GRIN2D O15399 1/20 0.34
GRIN3B O60391 1/20 0.34
GRIN1 Q05586 1/20 0.34
GRIN2A Q12879 1/20 0.34
GRIN2B Q13224 1/20 0.34
GRIN2C Q14957 1/20 0.34
GRIN3A Q8TCU5 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7995094 0.92 ALDH1A1 (0.36) GAAMAPTPRCPMTNR1AMTNR1B
SCHEMBL6831393 0.80 HTR2A (0.36) MTNR1AMTNR1BALDH1A1OPRM1OPRK1
SCHEMBL10505998 0.75 MAPT (0.47) GAAMAPTPRCPMTNR1AMTNR1B
SCHEMBL28873839 0.75 GAA (0.39) GAAMAPTGRIN2DGRIN3BGRIN1
SCHEMBL7099613 0.74 GAA (0.36) GAAMAPTMAPK1GRIN2DGRIN3B
SCHEMBL30488180 0.72 ALDH1A1 (0.39) GAAMTNR1AMTNR1BTSHRMEN1
SCHEMBL9631444 0.70 MAPT (0.47) GAAMAPTTSHRGRIN2DGRIN3B
SCHEMBL5319112 0.69 SLC22A1 (0.50) GAAMAPTPRCPMEN1KMT2A
SCHEMBL3249767 0.69 CYP2D6 (0.41) GAAMAPTTSHRMEN1KMT2A
SCHEMBL3240481 0.68 PDE5A (0.37) TSHRMEN1KMT2AALDH1A1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109790125-B Tetrahydroisoquinoline kappa opioid antagonists 研究三角协会 2022-07-05 CN claimed
CN-109790125-B Tetrahydroisoquinoline kappa opioid antagonists 研究三角协会 2022-07-05 CN disclosed
CN-109776414-A A kind of Bcl-2 protein inhibitor and its preparation method and application 山东大学 2019-05-21 CN disclosed