SCHEMBL5740276

SCHEMBL5740276

COC(=O)Oc1cn2ncnc(Nc3cc[nH]n3)c2c1C

nearest known ligand 0.43

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
KDR P35968 10/20 0.43
MAPK14 Q16539 10/20 0.41
EGFR P00533 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14451965 0.90 KDR (0.42) KDRMAPK14EGFR
SCHEMBL5741796 0.84 KDR (0.44) KDRMAPK14
SCHEMBL5741996 0.83 KDR (0.42) KDRMAPK14
SCHEMBL1461269 0.83 KDR (0.62) KDRMAPK14
SCHEMBL27561534 0.81 KDR (0.50) KDRMAPK14
SCHEMBL5740473 0.80 MAP2K1 (0.52) KDRMAPK14EGFR
SCHEMBL5740103 0.79 KDR (0.59) KDRMAPK14EGFR
SCHEMBL5738800 0.78 KDR (0.48) KDRMAPK14EGFR
SCHEMBL5740776 0.78 KDR (0.53) KDRMAPK14EGFR
SCHEMBL5741836 0.78 KDR (0.72) KDREGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1183033-B1 PYRROLOTRIAZINE INHIBITORS OF KINASES BRISTOL MYERS SQUIBB CO (US) 2006-03-01 EP claimed