SCHEMBL5741796

SCHEMBL5741796

COC(=O)Oc1cn2ncnc(Nc3cc(C)[nH]n3)c2c1C

nearest known ligand 0.44

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
KDR P35968 9/20 0.44
MAPK14 Q16539 10/20 0.40
AURKA O14965 1/20 0.39
AURKB Q96GD4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5740276 0.84 KDR (0.43) KDRMAPK14
SCHEMBL4050114 0.83 KDR (0.60) KDRMAPK14
SCHEMBL14469942 0.80 KDR (0.43) KDRMAPK14
SCHEMBL5741996 0.80 KDR (0.42) KDRMAPK14
SCHEMBL6112565 0.78 MAP2K1 (0.59) KDRMAPK14
SCHEMBL5740103 0.78 KDR (0.59) KDRMAPK14
SCHEMBL5740776 0.77 KDR (0.53) KDRMAPK14
SCHEMBL5739989 0.77 KDR (0.53) KDRMAPK14
SCHEMBL5740473 0.77 MAP2K1 (0.52) KDRMAPK14
SCHEMBL5739719 0.76 KDR (0.57) KDRMAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1183033-B1 PYRROLOTRIAZINE INHIBITORS OF KINASES BRISTOL MYERS SQUIBB CO (US) 2006-03-01 EP claimed