SCHEMBL5740293

SCHEMBL5740293

CCOC(=O)Oc1cn2ncnc(Nc3ccc(OC)nc3)c2c1C

nearest known ligand 0.49

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MAP2K1 Q02750 1/20 0.49
KDR P35968 13/20 0.47
EGFR P00533 3/20 0.44
ERBB2 P04626 3/20 0.44
MAPK14 Q16539 3/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5739638 0.92 KDR (0.48) MAP2K1KDREGFRMAPK14
SCHEMBL5740449 0.92 KDR (0.49) MAP2K1KDREGFRERBB2
SCHEMBL5740887 0.91 EGFR (0.50) MAP2K1KDREGFRERBB2MAPK14
SCHEMBL14451959 0.88 KDR (0.48) MAP2K1KDREGFRMAPK14
SCHEMBL4044547 0.85 MAP2K1 (0.67) MAP2K1KDREGFRERBB2MAPK14
SCHEMBL5740347 0.84 EGFR (0.46) MAP2K1KDREGFRERBB2
SCHEMBL5738887 0.81 KDR (0.46) MAP2K1KDREGFRMAPK14
SCHEMBL4053673 0.80 KDR (0.68) MAP2K1KDREGFRERBB2MAPK14
SCHEMBL7600802 0.80 KDR (0.57) MAP2K1KDREGFRERBB2MAPK14
SCHEMBL5522435 0.80 KDR (0.62) MAP2K1KDREGFRERBB2MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1183033-B1 PYRROLOTRIAZINE INHIBITORS OF KINASES BRISTOL MYERS SQUIBB CO (US) 2006-03-01 EP claimed