SCHEMBL5740347

SCHEMBL5740347

CCc1c(OC(=O)OC)cn2ncnc(Nc3ccc(OC)nc3)c12

nearest known ligand 0.46

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
EGFR P00533 13/20 0.46
ERBB2 P04626 13/20 0.46
KDR P35968 6/20 0.44
MAP2K1 Q02750 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5740887 0.94 EGFR (0.50) EGFRERBB2KDRMAP2K1
SCHEMBL5740924 0.92 EGFR (0.48) EGFRERBB2KDRMAP2K1
SCHEMBL5739638 0.87 KDR (0.48) EGFRKDRMAP2K1
SCHEMBL4049775 0.84 EGFR (0.58) EGFRERBB2KDRMAP2K1
SCHEMBL4051995 0.84 EGFR (0.58) EGFRERBB2KDR
SCHEMBL5740293 0.84 MAP2K1 (0.49) EGFRERBB2KDRMAP2K1
SCHEMBL5740449 0.83 KDR (0.49) EGFRERBB2KDRMAP2K1
SCHEMBL5516129 0.82 EGFR (0.68) EGFRERBB2KDRMAP2K1
SCHEMBL5739484 0.81 EGFR (0.54) EGFRERBB2KDRMAP2K1
SCHEMBL5741555 0.81 EGFR (0.59) EGFRERBB2KDRMAP2K1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1183033-B1 PYRROLOTRIAZINE INHIBITORS OF KINASES BRISTOL MYERS SQUIBB CO (US) 2006-03-01 EP claimed