SCHEMBL5740912

SCHEMBL5740912

CC(=O)ON(C(c1cccc(C(F)(F)F)c1)S(=O)(=O)c1ccc(Br)cc1)C(C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.39
CES2 O00748 2/20 0.38
DDR1 Q08345 1/20 0.37
ADAMTS4 O75173 1/20 0.36
MMP13 P45452 1/20 0.36
LMNA P02545 2/20 0.36
ALDH1A1 P00352 1/20 0.36
NPSR1 Q6W5P4 4/20 0.36
SLC6A4 P31645 2/20 0.35
HTR2C P28335 1/20 0.35
HTR2B P41595 1/20 0.35
HTR6 P50406 1/20 0.35
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
GAA P10253 1/20 0.34
CNR2 P34972 1/20 0.34
EPAS1 Q99814 1/20 0.34
IGF1R P08069 1/20 0.33
HTT P42858 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5740920 0.78 MAPT (0.41) MAPTCES2DDR1ADAMTS4MMP13
SCHEMBL381808 0.73 ACP3 (0.43) CES2MMP13LMNAALDH1A1NPSR1
SCHEMBL5259685 0.70 NPSR1 (0.43) MAPTCES2DDR1ADAMTS4MMP13
SCHEMBL27762553 0.65 CES2 (0.49) CES2LMNAALDH1A1NPSR1MEN1
SCHEMBL3077103 0.63 CES2 (0.50) CES2ADAMTS4MMP13LMNANPSR1
SCHEMBL9237550 0.63 CES2 (0.47) MAPTCES2LMNAALDH1A1NPSR1
SCHEMBL330908 0.63 CES2 (0.53) CES2ALDH1A1NPSR1MEN1KMT2A
SCHEMBL6915011 0.62 CYP3A4 (0.45) CES2ADAMTS4MMP13LMNAALDH1A1
SCHEMBL4749525 0.62 CES2 (0.46) MAPTCES2LMNAALDH1A1NPSR1
SCHEMBL3458826 0.62 CES2 (0.55) CES2ALDH1A1NPSR1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1620422-A2 PHENYL SUBSTITUTED CARBOXYLIC ACIDS AS INHIBITORS OF PROTEIN TYROSINE PHOSPHATASE-1B The Institutes for Pharmaceutical Discovery, LLC (US) 2006-02-01 EP disclosed
WO-2004099170-A2 PHENYL SUBSTITUTED CARBOXYLIC ACIDS AS INHIBITORS OF PROTEIN TYROSINE PHOSPHATASE-1B THE INSTITUTES FOR PHARMACEUTICAL DISCOVERY, LLC (US) 2004-11-18 WO disclosed