SCHEMBL5741832

SCHEMBL5741832

COc1ccccc1-c1cc(Nc2ccc3nc(-c4cccc(F)c4)cc(N)c3c2)nc(N)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AGPAT2 O15120 5/20 0.46
TP53 P04637 3/20 0.44
MAPT P10636 3/20 0.44
ALOX15 P16050 2/20 0.44
HSD17B10 Q99714 2/20 0.44
TSHR P16473 2/20 0.44
HPGD P15428 1/20 0.44
MAPK1 P28482 1/20 0.44
HTT P42858 1/20 0.44
KMT2A Q03164 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
USP2 O75604 2/20 0.44
LMNA P02545 2/20 0.44
CYP1A2 P05177 2/20 0.44
CYP2D6 P10635 2/20 0.44
CYP2C19 P33261 2/20 0.44
ALDH1A1 P00352 1/20 0.44
CLK4 Q9HAZ1 1/20 0.44
HSP90AA1 P07900 2/20 0.42
HSP90AB1 P08238 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5740482 0.92 ALOX15 (0.48) AGPAT2TP53MAPTALOX15HSD17B10
SCHEMBL5741860 0.92 MAPT (0.52) AGPAT2TP53MAPTALOX15HSD17B10
SCHEMBL5743121 0.90 AGPAT2 (0.55) AGPAT2TP53MAPTALOX15HSD17B10
SCHEMBL5741949 0.89 TP53 (0.49) AGPAT2TP53MAPTALOX15HSD17B10
SCHEMBL5744254 0.88 AGPAT2 (0.46) AGPAT2ROCK2ABCG2CYP3A4AURKA
SCHEMBL5742032 0.88 AGPAT2 (0.46) AGPAT2ROCK2ABCG2CYP3A4AURKA
SCHEMBL5740131 0.88 AGPAT2 (0.54) AGPAT2TP53MAPTALOX15HSD17B10
SCHEMBL5743044 0.88 AGPAT2 (0.50) AGPAT2TP53MAPTLMNAROCK2
SCHEMBL5741121 0.87 ABCG2 (0.47) AGPAT2TP53MAPTALOX15HSD17B10
SCHEMBL5743021 0.87 AGPAT2 (0.46) AGPAT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1339706-B1 N-TYPE CALCIUM CHANNEL ANTAGONISTS FOR THE TREATMENT OF PAIN ASTRAZENECA AB (SE) 2006-04-19 EP disclosed