SCHEMBL5742553

SCHEMBL5742553

Cc1cc(Nc2ccc3nc(C)cc(N)c3c2)nc(N)n1

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DOT1L Q8TEK3 4/20 0.78
TERT O14746 7/20 0.72
CYP1A2 P05177 2/20 0.61
CYP2D6 P10635 1/20 0.61
RAB9A P51151 2/20 0.58
NPC1 O15118 1/20 0.58
CYP3A4 P08684 1/20 0.58
CYP2C19 P33261 1/20 0.58
GNG2 P59768 2/20 0.58
GNB1 P62873 2/20 0.58
MEN1 O00255 1/20 0.58
MMP1 P03956 1/20 0.58
MMP9 P14780 1/20 0.58
ALOX15 P16050 1/20 0.58
BLM P54132 1/20 0.58
KMT2A Q03164 1/20 0.58
RAC1 P63000 2/20 0.55
MAPT P10636 2/20 0.53
ROCK2 O75116 1/20 0.51
DNMT1 P26358 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13039513 0.86 DOT1L (0.74) DOT1LTERTCYP1A2RAB9ANPC1
SCHEMBL5744090 0.86 DOT1L (0.59) DOT1LTERTCYP1A2CYP2D6RAB9A
SCHEMBL5741763 0.86 DOT1L (0.62) DOT1LTERTCYP1A2CYP2D6GNG2
SCHEMBL13305664 0.83 DOT1L (0.90) DOT1LTERTGNG2GNB1MEN1
SCHEMBL5742678 0.83 AGPAT2 (0.61) DOT1LTERTCYP1A2RAB9ANPC1
SCHEMBL4074842 0.82 TERT (0.91) DOT1LTERTGNG2GNB1MEN1
SCHEMBL5741412 0.81 DOT1L (0.57) DOT1LTERTCYP1A2CYP2D6GNG2
SCHEMBL27890181 0.81 TERT (0.69) DOT1LTERTGNG2GNB1MEN1
SCHEMBL5740573 0.81 DOT1L (0.57) DOT1LTERTMAPT
SCHEMBL5742405 0.81 DOT1L (0.56) DOT1LTERTCYP1A2CYP2D6GNG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1339706-B1 N-TYPE CALCIUM CHANNEL ANTAGONISTS FOR THE TREATMENT OF PAIN ASTRAZENECA AB (SE) 2006-04-19 EP disclosed