SCHEMBL5742787

SCHEMBL5742787

CC(C)(C)OC(=O)ON1CCC2C(=O)CCCC21

nearest known ligand 0.33

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PREP P48147 2/20 0.32
HPGD P15428 1/20 0.31
CHRM2 P08172 1/20 0.31
CHRM1 P11229 1/20 0.31
CHRM3 P20309 1/20 0.31
DDB1 Q16531 1/20 0.30
CRBN Q96SW2 1/20 0.30
KDM4E B2RXH2 1/20 0.30
MAPT P10636 1/20 0.30
THRB P10828 1/20 0.30
EPHX1 P07099 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1691897 0.77 HSD11B1 (0.40) PREPHPGDCHRM2CHRM1CHRM3
SCHEMBL1691937 0.77 HSD11B1 (0.40) PREPHPGDCHRM2CHRM1CHRM3
SCHEMBL5938430 0.73 HSD11B1 (0.46)
SCHEMBL5939353 0.73 HSD11B1 (0.46)
SCHEMBL1692175 0.73 ALDH1A1 (0.33)
SCHEMBL3383542 0.71 DDB1 (0.33) DDB1CRBNKDM4EMAPTTHRB
SCHEMBL23406491 0.70 HSD11B1 (0.41) HPGDCHRM2CHRM1CHRM3DDB1
SCHEMBL5938275 0.70 HSD11B1 (0.41) HPGDCHRM2CHRM1CHRM3DDB1
SCHEMBL23406490 0.70 HSD11B1 (0.41) HPGDCHRM2CHRM1CHRM3DDB1
SCHEMBL15245630 0.69 HSD11B1 (0.42) HPGDEPHX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1453512-B1 ACETYLENE DERIVATIVES HAVING MGLUR 5 ANTAGONISTIC ACTIVITY NOVARTIS AG (CH) 2006-05-31 EP claimed