SCHEMBL5742820

SCHEMBL5742820

CSc1nc(NCc2ccc(C(N)=O)c(-c3ccccc3N)c2)cc(-c2cccnc2)n1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 8/20 0.65
VCP P55072 1/20 0.42
MKNK1 Q9BUB5 1/20 0.40
MKNK2 Q9HBH9 1/20 0.40
PTGDR Q13258 1/20 0.40
CYP3A4 P08684 3/20 0.39
HDAC3 O15379 1/20 0.39
NCOR1 O75376 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC11 Q96DB2 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
NCOR2 Q9Y618 1/20 0.39
ALDH1A1 P00352 2/20 0.39
CYP1A2 P05177 2/20 0.39
CYP2D6 P10635 2/20 0.39
HSD17B10 Q99714 2/20 0.39
CLK4 Q9HAZ1 1/20 0.39
BACE1 P56817 1/20 0.39
KDM4E B2RXH2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30518168 0.81 HDAC1 (0.60) HDAC1CYP3A4HDAC3NCOR1HDAC2
SCHEMBL210054 0.79 HDAC1 (1.00) HDAC1CYP3A4HDAC3NCOR1HDAC2
SCHEMBL213325 0.77 HDAC1 (0.71) HDAC1VCPMKNK1MKNK2PTGDR
SCHEMBL18808254 0.76 HDAC1 (0.72) HDAC1VCPCYP3A4HDAC3NCOR1
SCHEMBL5733996 0.71 HDAC1 (0.48) HDAC1MKNK2CYP3A4HDAC3NCOR1
SCHEMBL27836360 0.69 HDAC1 (0.59) HDAC1CYP3A4HDAC3HDAC2HDAC11
SCHEMBL14917848 0.67 HDAC1 (0.61) HDAC1HDAC8HDAC6
SCHEMBL167082 0.66 BCAT2 (0.67) MKNK1MKNK2
SCHEMBL31227976 0.66 BCAT2 (0.67) MKNK1MKNK2
SCHEMBL30514275 0.66 BCAT2 (0.67) MKNK1MKNK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1735319-A1 INHIBITORS OF HISTONE DEACETYLASE Methylgene, Inc. (CA) 2006-12-27 EP claimed
WO-2005092899-A1 INHIBITORS OF HISTONE DEACETYLASE METHYLGENE INC. (CA) 2005-10-06 WO claimed