SCHEMBL5733996

SCHEMBL5733996

NC(=O)c1ccc(CNc2nccc(-c3ccncc3)n2)cc1-c1ccccc1N

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 13/20 0.48
HDAC3 O15379 5/20 0.48
NCOR1 O75376 5/20 0.48
HDAC2 Q92769 4/20 0.48
HDAC8 Q9BY41 2/20 0.48
HDAC6 Q9UBN7 2/20 0.48
CYP3A4 P08684 1/20 0.48
HDAC11 Q96DB2 1/20 0.48
NCOR2 Q9Y618 1/20 0.48
CDC7 O00311 2/20 0.46
ROCK2 O75116 2/20 0.46
MAP4K4 O95819 2/20 0.46
GSK3B P49841 2/20 0.46
CLK4 Q9HAZ1 2/20 0.46
MKNK2 Q9HBH9 1/20 0.46
HDAC4 P56524 1/20 0.45
MEF2D Q14814 1/20 0.45
PIM1 P11309 1/20 0.42
CDK2 P24941 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30518168 0.90 HDAC1 (0.60) HDAC1HDAC3NCOR1HDAC2HDAC8
SCHEMBL210559 0.74 HDAC1 (0.82) HDAC1HDAC3NCOR1HDAC2HDAC8
SCHEMBL5091711 0.72 MAPK8 (0.55) HDAC1HDAC3NCOR1HDAC2HDAC8
SCHEMBL5742820 0.71 HDAC1 (0.65) HDAC1HDAC3NCOR1HDAC2HDAC8
SCHEMBL6648686 0.70 CAMKK2 (0.67) GSK3B
SCHEMBL7464625 0.69 DYRK1A (0.52) HDAC1HDAC3NCOR1HDAC2HDAC8
SCHEMBL5094681 0.69 MAPK8 (0.54) HDAC1HDAC3NCOR1HDAC2HDAC8
SCHEMBL212828 0.69 PDE4B (0.44) HDAC1HDAC3
SCHEMBL27576350 0.68 CAMKK2 (0.55) HDAC1HDAC3NCOR1HDAC2HDAC8
SCHEMBL2732829 0.67 HDAC1 (0.85) HDAC1HDAC3NCOR1HDAC2HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1735319-A1 INHIBITORS OF HISTONE DEACETYLASE Methylgene, Inc. (CA) 2006-12-27 EP claimed
WO-2005092899-A1 INHIBITORS OF HISTONE DEACETYLASE METHYLGENE INC. (CA) 2005-10-06 WO claimed