SCHEMBL5742833

SCHEMBL5742833

CCCCCc1cc(Nc2ccc3nc(-c4ccc(Cl)cc4)cc(N)c3c2)nc(N)n1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 6/20 0.48
AGPAT2 O15120 5/20 0.48
NPC1 O15118 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C19 P33261 1/20 0.41
RAB9A P51151 1/20 0.41
TERT O14746 1/20 0.41
HRH2 P25021 1/20 0.40
HRH3 Q9Y5N1 1/20 0.40
DOT1L Q8TEK3 2/20 0.40
OPRL1 P41146 1/20 0.39
TP53 P04637 1/20 0.39
MAPT P10636 1/20 0.39
ASIC3 Q9UHC3 1/20 0.38
TLR8 Q9NR97 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5742344 0.90 MCHR1 (0.44) MCHR1AGPAT2TERTHRH2HRH3
SCHEMBL5740235 0.90 MCHR1 (0.44) MCHR1AGPAT2TERTDOT1LTLR8
SCHEMBL5742308 0.88 AGPAT2 (0.53) MCHR1AGPAT2ASIC3TLR8
SCHEMBL5743256 0.80 MCHR1 (0.59) MCHR1AGPAT2TLR8
SCHEMBL5740139 0.80 AGPAT2 (0.60) AGPAT2NPC1CYP1A2CYP3A4CYP2C19
SCHEMBL5743347 0.79 AGPAT2 (0.57) AGPAT2NPC1CYP1A2CYP3A4CYP2C19
SCHEMBL5742678 0.79 AGPAT2 (0.61) AGPAT2NPC1CYP1A2CYP3A4CYP2C19
SCHEMBL5742169 0.78 MCHR1 (0.44) MCHR1AGPAT2TERTDOT1LTP53
SCHEMBL5744288 0.78 KDM4E (0.56) MCHR1AGPAT2NPC1CYP1A2CYP3A4
SCHEMBL5742888 0.78 AGPAT2 (0.64) AGPAT2NPC1CYP1A2CYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1339706-B1 N-TYPE CALCIUM CHANNEL ANTAGONISTS FOR THE TREATMENT OF PAIN ASTRAZENECA AB (SE) 2006-04-19 EP disclosed