SCHEMBL5743484

SCHEMBL5743484

COc1cccc(Cc2ncc(C=O)c3cc(OC4CCCC4)c(OC)cc23)c1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.42
PDE4A P27815 7/20 0.42
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
PDE4B Q07343 6/20 0.41
PDE4D Q08499 6/20 0.41
PDE4C Q08493 5/20 0.41
ADRA1A P35348 1/20 0.40
HRH1 P35367 1/20 0.40
HRH3 Q9Y5N1 1/20 0.40
KIT P10721 1/20 0.39
POLB P06746 1/20 0.39
ALPL P05186 1/20 0.39
HTT P42858 1/20 0.39
NMT1 P30419 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5745797 0.82 ERN1 (0.46) ALDH1A1ADRA1AKITHTT
SCHEMBL5745105 0.82 ERN1 (0.46) ALDH1A1ADRA1AKITHTT
SCHEMBL5744687 0.82 ERN1 (0.42) ALDH1A1MEN1KMT2ANPSR1POLB
SCHEMBL5745438 0.81 PDE10A (0.42) ADRA1AKITHTT
SCHEMBL5743598 0.80 DHFR (0.44) ALDH1A1PDE4ANPSR1PDE4BPDE4D
SCHEMBL5745922 0.79 PDE4B (0.49) PDE4AMEN1KMT2APDE4BPDE4D
SCHEMBL5743602 0.77 PDE10A (0.41) HTT
SCHEMBL5744723 0.76 DHFR (0.38) ALDH1A1PDE4ANPSR1PDE4BPDE4D
SCHEMBL5746367 0.75 DPP4 (0.41) ALDH1A1MEN1KMT2APDE4D
SCHEMBL5745200 0.75 PDE10A (0.39) ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7067529-B2 Glutamine fructose-y-phosphate amidotransferase (GFAT) inhibitors HOFFMANN-LA ROCHE INC. (US) 2006-06-27 US disclosed
EP-1631551-A2 ISOQUINOLINE DERIVATIVES AND THEIR USE AS GFAT INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2006-03-08 EP disclosed
US-20040259910-A1 Glutamine fructose-y-phosphate amidotransferase (GFAT) inhibitors BOLIN DAVID ROBERT (US) 2004-12-23 US disclosed
WO-2004101528-A2 ISOQUINOLINE DERIVATIVES AND THEIR USE AS GFAT INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2004-11-25 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040259910-A1 Glutamine fructose-y-phosphate amidotransferase (GFAT) inhibitors GFPT1, GLS2, GLS ALDH1A1 1211/4885PDE4A 2228/4885MEN1 2407/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.