SCHEMBL5744591

SCHEMBL5744591

O=C1CC(C(=O)N2CCC(O)(c3ccccc3)CC2)N(C(=O)c2ccc(-c3cccnc3)cc2)C1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.53
LMNA P02545 2/20 0.53
MKNK1 Q9BUB5 2/20 0.44
MKNK2 Q9HBH9 2/20 0.44
AVPR2 P30518 1/20 0.44
OXTR P30559 1/20 0.44
AVPR1A P37288 1/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
PKM P14618 1/20 0.43
CNR2 P34972 1/20 0.42
ABL1 P00519 3/20 0.41
BCR P11274 3/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA7 P43166 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5744595 1.00 ALDH1A1 (0.53) ALDH1A1LMNAMKNK1MKNK2AVPR2
SCHEMBL5741756 0.92 CA12 (0.47) ALDH1A1LMNAMEN1KMT2ACA12
SCHEMBL5741758 0.92 CA12 (0.47) ALDH1A1LMNAMEN1KMT2ACA12
SCHEMBL5745769 0.92 ALDH1A1 (0.48) ALDH1A1LMNAMEN1KMT2APKM
SCHEMBL5745771 0.92 ALDH1A1 (0.48) ALDH1A1LMNAMEN1KMT2APKM
SCHEMBL4936043 0.86 OXTR (0.49) ALDH1A1LMNAMKNK1MKNK2AVPR2
SCHEMBL4936051 0.86 OXTR (0.49) ALDH1A1LMNAMKNK1MKNK2AVPR2
SCHEMBL5742550 0.78 MKNK1 (0.46) ALDH1A1MKNK1MKNK2AVPR2OXTR
SCHEMBL5742548 0.78 MKNK1 (0.46) ALDH1A1MKNK1MKNK2AVPR2OXTR
SCHEMBL4943212 0.77 OXTR (0.49) ALDH1A1LMNAOXTRAVPR1AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1268419-B1 PYRROLIDINE DERIVATIVES USEFUL AS BAX INHIBITORS APPLIED RESEARCH SYSTEMS (AN) 2006-06-21 EP claimed