SCHEMBL5745193

SCHEMBL5745193

CN(C)CCCOc1cccc2oc3ccccc3c12

nearest known ligand 0.61

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HTR1B P28222 3/20 0.61
HRH1 P35367 1/20 0.48
ADRB2 P07550 1/20 0.47
HTT P42858 1/20 0.44
MAOA P21397 1/20 0.43
HTR7 P34969 1/20 0.43
SIGMAR1 Q99720 1/20 0.43
BCHE P06276 1/20 0.42
ACHE P22303 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5748560 0.93 HTR1B (0.60) HTR1BADRB2HTTMAOAHTR7
SCHEMBL5749134 0.89 MAOA (0.59) HTR1BMAOABCHEACHE
SCHEMBL5748254 0.86 XDH (0.57) HTR1BADRB2BCHEACHE
SCHEMBL11843761 0.85 XDH (0.51) HTR1BSIGMAR1BCHEACHE
SCHEMBL12967977 0.83 CDC25A (0.52) HTR1BADRB2MAOA
SCHEMBL5745354 0.82 MAOA (0.61) HTR1BHTTMAOAHTR7BCHE
SCHEMBL15473271 0.81 CYP2A6 (0.59) HTR1BADRB2MAOA
SCHEMBL10431487 0.81 ADRB2 (0.48) HTR1BHRH1ADRB2HTTMAOA
SCHEMBL5748059 0.81 POLB (0.53) HTR1BADRB2
SCHEMBL5747324 0.80 HTR1B (0.58) HTR1BHRH1ADRB2MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1711463-A2 AMINO-SUBSTITUTED TRICYCLIC DERIVATIVES AND METHODS OF USE ABBOTT LABORATORIES (US) 2006-10-18 EP disclosed
WO-2005077899-A2 AMINO-SUBSTITUTED TRICYCLIC DERIVATIVES AND METHODS OF USE ABBOTT LABORATORIES (US) 2005-08-25 WO disclosed