SCHEMBL5745856

SCHEMBL5745856

CCCNCCOc1cccc2c1[C@@H](O)c1ccccc1-2

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR1B P28222 3/20 0.53
KDM4E B2RXH2 8/20 0.49
ADRB2 P07550 4/20 0.48
SMN1; SMN2 Q16637 5/20 0.44
HTT P42858 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.43
ALDH1A1 P00352 3/20 0.43
HTR1A P08908 2/20 0.41
ADRA1D P25100 2/20 0.41
ADRA1A P35348 2/20 0.41
ADRA1B P35368 2/20 0.41
HTR1D P28221 1/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
GAA P10253 1/20 0.40
ADRB1 P08588 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5747826 0.91 ADRB2 (0.59) HTR1BKDM4EADRB2SMN1; SMN2HTT
SCHEMBL5744105 0.87 ADRB2 (0.55) HTR1BKDM4EADRB2SMN1; SMN2HTT
SCHEMBL5746575 0.85 KDM4E (0.55) HTR1BKDM4EADRB2SMN1; SMN2HTT
SCHEMBL5746987 0.84 HRH1 (0.51) HTR1BKDM4EADRB2L3MBTL1ALDH1A1
SCHEMBL5747675 0.78 HTR1B (0.46) HTR1BKDM4ESMN1; SMN2ALDH1A1MEN1
SCHEMBL5747194 0.77 KDM4E (0.52) HTR1BKDM4ESMN1; SMN2HTTALDH1A1
SCHEMBL5746581 0.73 HRH3 (0.61) KDM4ESMN1; SMN2HTTL3MBTL1ALDH1A1
SCHEMBL1795532 0.72 DRD2 (0.43) HTR1BKDM4EADRB2SMN1; SMN2ALDH1A1
SCHEMBL5748910 0.72 HRH3 (0.63) KDM4ESMN1; SMN2HTTL3MBTL1ALDH1A1
SCHEMBL5746264 0.72 ALDH1A1 (0.54) KDM4ESMN1; SMN2HTTL3MBTL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1711463-A2 AMINO-SUBSTITUTED TRICYCLIC DERIVATIVES AND METHODS OF USE ABBOTT LABORATORIES (US) 2006-10-18 EP claimed
WO-2005077899-A2 AMINO-SUBSTITUTED TRICYCLIC DERIVATIVES AND METHODS OF USE ABBOTT LABORATORIES (US) 2005-08-25 WO claimed
EP-1711463-A2 AMINO-SUBSTITUTED TRICYCLIC DERIVATIVES AND METHODS OF USE ABBOTT LABORATORIES (US) 2006-10-18 EP disclosed
WO-2005077899-A2 AMINO-SUBSTITUTED TRICYCLIC DERIVATIVES AND METHODS OF USE ABBOTT LABORATORIES (US) 2005-08-25 WO disclosed