SCHEMBL5746787

SCHEMBL5746787

Cc1cc(F)ccc1C1C2CNCC2CN1C(=O)OCc1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 1/20 0.46
POLB P06746 1/20 0.40
PDK1 Q15118 1/20 0.39
PDK2 Q15119 1/20 0.39
PDK3 Q15120 1/20 0.39
PDK4 Q16654 1/20 0.39
PKM P14618 1/20 0.39
PTGDR2 Q9Y5Y4 1/20 0.38
PARP1 P09874 1/20 0.37
SIGMAR1 Q99720 3/20 0.37
TMEM97 Q5BJF2 2/20 0.37
NPSR1 Q6W5P4 2/20 0.37
MRGPRX4 Q96LA9 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6317296 0.84 DRD2 (0.41) POLBPTGDR2SIGMAR1TMEM97
SCHEMBL5745277 0.83 TACR1 (0.39) HTR2C
SCHEMBL5746790 0.76 PTGDR2 (0.41) HTR2CPOLBPKMPTGDR2SIGMAR1
SCHEMBL6311280 0.76 DRD2 (0.40) HTR2CPOLBPKMSIGMAR1TMEM97
SCHEMBL5744862 0.75 CYP2D6 (0.41) POLBPKMPTGDR2
SCHEMBL4026871 0.74 HTR2C (0.42) HTR2CPDK1PDK2PDK3PDK4
SCHEMBL4027421 0.73 SMN1; SMN2 (0.43) HTR2CPKMPTGDR2SIGMAR1TMEM97
SCHEMBL2488624 0.73 PARP1 (0.46) PKMPTGDR2PARP1SIGMAR1TMEM97
SCHEMBL4024932 0.73 SMN1; SMN2 (0.43) HTR2CPKMPTGDR2SIGMAR1TMEM97
SCHEMBL4859941 0.73 PARP1 (0.46) PKMPTGDR2PARP1SIGMAR1TMEM97

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1638935-A1 NK1 ANTAGONIST Pfizer Products Inc. (US) 2006-03-29 EP disclosed
WO-2004110996-A1 NK1 ANTAGONIST PFIZER PRODUCTS INC. (US) 2004-12-23 WO disclosed