SCHEMBL5744862

SCHEMBL5744862

Cc1cc(F)ccc1C1C2C(=O)N(Cc3ccccc3)C(=O)C2CN1C(=O)OCc1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.41
ALDH1A1 P00352 2/20 0.39
LMNA P02545 1/20 0.39
PTGDR2 Q9Y5Y4 1/20 0.39
CYP3A4 P08684 2/20 0.38
TSHR P16473 2/20 0.38
MAPT P10636 1/20 0.38
CYP2C9 P11712 2/20 0.38
POLB P06746 1/20 0.38
PKM P14618 1/20 0.38
CACNA1G O43497 1/20 0.38
CACNA1H O95180 1/20 0.38
CACNA1I Q9P0X4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6309596 0.89 CACNA1G (0.43) CYP2D6ALDH1A1MAPTCACNA1GCACNA1H
SCHEMBL6319094 0.81 ALDH1A1 (0.45) CYP2D6ALDH1A1CYP3A4TSHRCYP2C9
SCHEMBL6311280 0.81 DRD2 (0.40) POLBPKMCACNA1GCACNA1HCACNA1I
SCHEMBL6317296 0.78 DRD2 (0.41) PTGDR2POLBCACNA1GCACNA1HCACNA1I
SCHEMBL5746787 0.75 HTR2C (0.46) PTGDR2POLBPKM
SCHEMBL6317300 0.73 PTGDR2 (0.41) PTGDR2POLBCACNA1GCACNA1HCACNA1I
SCHEMBL4859941 0.72 PARP1 (0.46) PTGDR2PKM
SCHEMBL2488624 0.72 PARP1 (0.46) PTGDR2PKM
SCHEMBL4030829 0.71 PDK1 (0.43) PTGDR2POLB
SCHEMBL2490272 0.71 PKM (0.43) PTGDR2PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1638935-A1 NK1 ANTAGONIST Pfizer Products Inc. (US) 2006-03-29 EP disclosed
US-20050043354-A1 NK1 antagonist PFIZER INC 2005-02-24 US disclosed
WO-2004110996-A1 NK1 ANTAGONIST PFIZER PRODUCTS INC. (US) 2004-12-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050043354-A1 NK1 antagonist TACR2, TACR1, TAC3 CYP2D6 2419/4885ALDH1A1 2855/4885LMNA 3815/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.