SCHEMBL5747367

SCHEMBL5747367

Cn1c2ccccc2c2cccc(OCCN3CCCCC3)c21

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.56
TSHR P16473 1/20 0.55
CYP2D6 P10635 2/20 0.52
CYP2C19 P33261 2/20 0.52
CYP1A2 P05177 1/20 0.52
HSD17B10 Q99714 1/20 0.52
HRH3 Q9Y5N1 4/20 0.52
HTR2A P28223 4/20 0.52
HTR7 P34969 2/20 0.52
HTR6 P50406 2/20 0.52
POLB P06746 1/20 0.51
HRH1 P35367 3/20 0.50
DRD1 P21728 2/20 0.50
DRD4 P21917 2/20 0.50
DRD5 P21918 2/20 0.50
DRD3 P35462 2/20 0.50
DRD2 P14416 1/20 0.50
HTR2C P28335 2/20 0.49
HTR2B P41595 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5748859 0.99 TDP1 (0.57) TDP1TSHRCYP2D6CYP2C19CYP1A2
SCHEMBL11376119 0.90 TDP1 (0.51) TDP1TSHRCYP2D6CYP2C19CYP1A2
SCHEMBL5748094 0.90 CYP2D6 (0.55) TDP1CYP2D6CYP2C19CYP1A2HRH3
SCHEMBL11382220 0.89 TDP1 (0.52) TDP1TSHRCYP2D6CYP2C19CYP1A2
SCHEMBL5749161 0.80 TDP1 (0.51) TDP1TSHRCYP2D6CYP2C19CYP1A2
SCHEMBL5748798 0.79 HTR1B (0.53) TSHRHTR6
SCHEMBL5747101 0.79 TDP1 (0.52) TDP1TSHRCYP2D6CYP2C19CYP1A2
SCHEMBL5747516 0.78 HTR1B (0.54)
SCHEMBL5745919 0.78 TDP1 (0.51) TDP1TSHRCYP2D6CYP2C19CYP1A2
SCHEMBL14970486 0.77 HRH3 (0.81) TDP1TSHRHRH3HTR2AHTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1711463-A2 AMINO-SUBSTITUTED TRICYCLIC DERIVATIVES AND METHODS OF USE ABBOTT LABORATORIES (US) 2006-10-18 EP disclosed
WO-2005077899-A2 AMINO-SUBSTITUTED TRICYCLIC DERIVATIVES AND METHODS OF USE ABBOTT LABORATORIES (US) 2005-08-25 WO disclosed