SCHEMBL5748798

SCHEMBL5748798

Cn1c2ccccc2c2cccc(OCCN)c21

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1B P28222 3/20 0.53
ALKBH5 Q6P6C2 1/20 0.50
FTO Q9C0B1 1/20 0.50
KDM4E B2RXH2 2/20 0.49
GPR3 P46089 1/20 0.44
HTR6 P50406 1/20 0.42
KCNA3 P22001 1/20 0.42
MCL1 Q07820 1/20 0.41
TP53 P04637 1/20 0.41
MAPK1 P28482 1/20 0.41
RAB9A P51151 1/20 0.41
LIMK1 P53667 1/20 0.40
HPGD P15428 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
HSP90AA1 P07900 1/20 0.38
IDO1 P14902 1/20 0.38
MAPT P10636 2/20 0.38
LMNA P02545 1/20 0.38
TSHR P16473 1/20 0.38
HTT P42858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5747516 0.93 HTR1B (0.54) HTR1BALKBH5FTOKDM4EGPR3
SCHEMBL15466278 0.83 ALKBH5 (0.54) ALKBH5FTOKDM4EGPR3TP53
SCHEMBL5749824 0.82 HTR1B (0.57) HTR1BALKBH5FTOKDM4EGPR3
SCHEMBL5770352 0.81 HRH1 (0.58) HTR1BALKBH5FTOGPR3HTR6
SCHEMBL5747639 0.81 HTR1B (0.61) HTR1BALKBH5FTOGPR3HTR6
SCHEMBL5748859 0.80 TDP1 (0.57) HTR6TSHR
SCHEMBL5747747 0.80 HTR1B (0.56) HTR1BALKBH5FTOGPR3KCNA3
SCHEMBL5748021 0.80 HTR1B (0.50) HTR1BALKBH5FTOKDM4EGPR3
SCHEMBL5747367 0.79 TDP1 (0.56) HTR6TSHR
SCHEMBL5771872 0.79 HTR1B (0.60) HTR1BALKBH5FTOHTR6KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1711463-A2 AMINO-SUBSTITUTED TRICYCLIC DERIVATIVES AND METHODS OF USE ABBOTT LABORATORIES (US) 2006-10-18 EP disclosed
WO-2005077899-A2 AMINO-SUBSTITUTED TRICYCLIC DERIVATIVES AND METHODS OF USE ABBOTT LABORATORIES (US) 2005-08-25 WO disclosed