SCHEMBL5747685

SCHEMBL5747685

NCCCOSc1cccc2oc3ccccc3c(=O)c12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 6/20 0.45
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
GLA P06280 1/20 0.42
CYP3A4 P08684 1/20 0.42
MAPT P10636 1/20 0.42
HPGD P15428 1/20 0.42
PGAM1 P18669 1/20 0.42
CASP1 P29466 1/20 0.42
CASP7 P55210 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
HSD17B10 Q99714 1/20 0.42
KDM5A P29375 1/20 0.40
TOP2A P11388 1/20 0.39
MGAM O43451 1/20 0.38
GAA P10253 1/20 0.38
SI P14410 1/20 0.38
MGAM2 Q2M2H8 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2D6 P10635 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5747968 0.84 MAOA (0.45) MAOAKDM4EALDH1A1GLACYP3A4
SCHEMBL5747519 0.82 MAOA (0.43) MAOAKDM4EALDH1A1GLACYP3A4
SCHEMBL5749171 0.82 XDH (0.57) MAOAMAPTXDH
SCHEMBL5746335 0.81 XDH (0.58) XDH
SCHEMBL5748857 0.81 XDH (0.55) MEN1NPC1KMT2AXDH
SCHEMBL5750263 0.81 TOP2A (0.43) MAOAKDM4EALDH1A1GLACYP3A4
SCHEMBL5745622 0.81 MAOA (0.47) MAOAKDM4EALDH1A1GLACYP3A4
SCHEMBL5746038 0.81 MAOA (0.47) MAOAKDM4EALDH1A1GLACYP3A4
SCHEMBL5747754 0.80 XDH (0.59) KDM4EALDH1A1MAPTXDH
SCHEMBL5748332 0.79 XDH (0.51) MAOAKDM4EALDH1A1GLACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1711463-A2 AMINO-SUBSTITUTED TRICYCLIC DERIVATIVES AND METHODS OF USE ABBOTT LABORATORIES (US) 2006-10-18 EP claimed
WO-2005077899-A2 AMINO-SUBSTITUTED TRICYCLIC DERIVATIVES AND METHODS OF USE ABBOTT LABORATORIES (US) 2005-08-25 WO claimed
EP-1711463-A2 AMINO-SUBSTITUTED TRICYCLIC DERIVATIVES AND METHODS OF USE ABBOTT LABORATORIES (US) 2006-10-18 EP disclosed
WO-2005077899-A2 AMINO-SUBSTITUTED TRICYCLIC DERIVATIVES AND METHODS OF USE ABBOTT LABORATORIES (US) 2005-08-25 WO disclosed