SCHEMBL5749070

SCHEMBL5749070

CCNCCCOc1cccc2oc3ccccc3c(=O)c12

nearest known ligand 0.57

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAOA P21397 3/20 0.57
HTR1B P28222 1/20 0.52
NMT2 O60551 2/20 0.46
NMT1 P30419 2/20 0.46
TOP2A P11388 3/20 0.45
CYP2A6 P11509 1/20 0.44
MEN1 O00255 1/20 0.44
NPC1 O15118 1/20 0.44
KMT2A Q03164 1/20 0.44
ADRB2 P07550 3/20 0.43
ADRB1 P08588 1/20 0.43
ADRB3 P13945 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5749598 0.96 MAOA (0.58) MAOAHTR1BTOP2ACYP2A6MEN1
SCHEMBL5749002 0.91 MAOA (0.56) MAOAHTR1BNMT2NMT1TOP2A
SCHEMBL5749350 0.90 HTR1B (0.57) HTR1BNMT2NMT1KMT2AADRB2
SCHEMBL5748795 0.88 HTR1B (0.58) MAOAHTR1BTOP2ACYP2A6MEN1
SCHEMBL5748462 0.87 MAOA (0.59) MAOAHTR1BCYP2A6MEN1NPC1
SCHEMBL5749472 0.86 MAOA (0.61) MAOAHTR1BCYP2A6MEN1NPC1
SCHEMBL5748148 0.85 HTR1B (0.62) MAOAHTR1BNMT2NMT1CYP2A6
SCHEMBL28198664 0.84 MAOA (0.62) MAOATOP2ACYP2A6NPC1
SCHEMBL5749229 0.82 HTR1B (0.58) HTR1BNMT2NMT1CYP2A6ADRB2
SCHEMBL6893811 0.81 MAOA (0.69) MAOACYP2A6MEN1NPC1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1711463-A2 AMINO-SUBSTITUTED TRICYCLIC DERIVATIVES AND METHODS OF USE ABBOTT LABORATORIES (US) 2006-10-18 EP disclosed
WO-2005077899-A2 AMINO-SUBSTITUTED TRICYCLIC DERIVATIVES AND METHODS OF USE ABBOTT LABORATORIES (US) 2005-08-25 WO disclosed