SCHEMBL5749264

SCHEMBL5749264

c1ccc2c(c1)oc1cccc(OCCCN3CCCC3)c12

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.59
XDH P47989 2/20 0.58
HRH3 Q9Y5N1 8/20 0.56
HTR2A P28223 2/20 0.56
HTR7 P34969 2/20 0.56
HTR6 P50406 2/20 0.56
CYP2D6 P10635 2/20 0.56
CYP2C19 P33261 2/20 0.56
NMT2 O60551 1/20 0.55
NMT1 P30419 1/20 0.55
ALDH1A1 P00352 2/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
MAOB P27338 4/20 0.52
BCHE P06276 1/20 0.52
ACHE P22303 1/20 0.52
L3MBTL1 Q9Y468 2/20 0.51
HRH1 P35367 2/20 0.51
CYP1A2 P05177 1/20 0.51
DRD2 P14416 1/20 0.51
DRD1 P21728 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5749883 0.99 XDH (0.59) TDP1XDHHRH3HTR2AHTR7
SCHEMBL5744863 0.97 TDP1 (0.56) TDP1XDHHRH3HTR2AHTR7
SCHEMBL5747870 0.93 TDP1 (0.55) TDP1XDHHRH3HTR2AHTR7
SCHEMBL5748468 0.92 TSHR (0.56) TDP1XDHHRH3HTR2AHTR7
SCHEMBL28675845 0.90 XDH (0.66) TDP1XDHHRH3HTR2AHTR7
SCHEMBL5748656 0.83 XDH (0.58) TDP1XDHHRH3MAOBBCHE
SCHEMBL5748784 0.82 XDH (0.58) TDP1XDHHRH3HTR2AHTR7
SCHEMBL5747713 0.81 XDH (0.55) TDP1XDHHRH3MAOBBCHE
SCHEMBL10431487 0.78 ADRB2 (0.48) ALDH1A1SMN1; SMN2HRH1
SCHEMBL14970546 0.77 HRH3 (0.89) TDP1HRH3HTR2AHTR7HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1711463-A2 AMINO-SUBSTITUTED TRICYCLIC DERIVATIVES AND METHODS OF USE ABBOTT LABORATORIES (US) 2006-10-18 EP disclosed
WO-2005077899-A2 AMINO-SUBSTITUTED TRICYCLIC DERIVATIVES AND METHODS OF USE ABBOTT LABORATORIES (US) 2005-08-25 WO disclosed