SCHEMBL5749337

SCHEMBL5749337

Nc1c(C=O)ccc2cc3ccccc3cc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.41
HSD17B10 Q99714 3/20 0.41
HIF1A Q16665 2/20 0.41
TDP1 Q9NUW8 2/20 0.41
CYP3A4 P08684 2/20 0.41
ALOX15 P16050 1/20 0.41
CASP1 P29466 1/20 0.41
CASP7 P55210 1/20 0.41
HBB P68871 1/20 0.41
GAA P10253 4/20 0.41
KDM4E B2RXH2 3/20 0.41
CYP1B1 Q16678 1/20 0.39
ERN1 O75460 3/20 0.38
KMT2A Q03164 5/20 0.38
MEN1 O00255 4/20 0.38
LMNA P02545 2/20 0.38
THRB P10828 1/20 0.38
BLM P54132 1/20 0.38
PI4KA P42356 1/20 0.37
PI4K2B Q8TCG2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29950700 0.82 ERN1 (0.46) ALDH1A1HSD17B10TDP1CYP3A4CASP1
SCHEMBL514682 0.82 ERN1 (0.46) ALDH1A1HSD17B10TDP1CYP3A4CASP1
Hydrochloric Acid SCHEMBL27803975 0.81 ERN1 (0.44) ALDH1A1HSD17B10HIF1ATDP1CYP3A4
SCHEMBL347177 0.79 ERN1 (0.43) ALDH1A1HSD17B10HIF1ATDP1GAA
SCHEMBL545879 0.78 ERN1 (0.42) ALDH1A1HSD17B10HIF1ATDP1CYP3A4
SCHEMBL547776 0.78 ERN1 (0.42) ALDH1A1HSD17B10HIF1ATDP1CYP3A4
SCHEMBL984194 0.78 KMT2A (0.50) ALDH1A1HSD17B10HIF1ATDP1GAA
SCHEMBL39718 0.76 ALDH1A1 (0.50) ALDH1A1HSD17B10HIF1ATDP1CYP3A4
SCHEMBL29392367 0.76 ALDH1A1 (0.50) ALDH1A1HSD17B10HIF1ATDP1CYP3A4
SCHEMBL9851160 0.76 TYMS (0.45) ALDH1A1HSD17B10HIF1ATDP1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3044284-B1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2019-11-13 EP disclosed
US-9831448-B2 Metal complexes MERCK PATENT GMBH (DE) 2017-11-28 US disclosed
US-9831448-B2 Metal complexes MERCK PATENT GMBH (DE) 2017-11-28 US disclosed
US-20160233443-A1 Metal Complexes MERCK PATENT GMBH (DE) 2016-08-11 US disclosed
US-20160233443-A1 Metal Complexes MERCK PATENT GMBH (DE) 2016-08-11 US disclosed
WO-2015036074-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2015-03-19 WO disclosed
US-20060293503-A1 Polyaminopyridines and method for producing same SUMITOMO SEIKA CHEMICALS CO., LTD (JP) 2006-12-28 US disclosed
EP-1669390-A1 POLYAMINOPYRIDINES AND METHOD FOR PRODUCING SAME SUMITOMO SEIKA CHEMICALS CO., LTD. (JP) 2006-06-14 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160233443-A1 Metal Complexes AP1M1, SOD1, AP3M1 ALDH1A1 3771/4885HSD17B10 3051/4885HIF1A 4770/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.