SCHEMBL5750596

SCHEMBL5750596

CNCCCOc1cccc2c1c1ccccc1c(=O)n2C

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 3/20 0.53
SLC6A4 P31645 2/20 0.53
HTR1B P28222 5/20 0.48
HTR1D P28221 1/20 0.48
HTR6 P50406 1/20 0.44
KDM4E B2RXH2 3/20 0.42
ALDH1A1 P00352 2/20 0.42
HPGD P15428 2/20 0.42
HSD17B10 Q99714 2/20 0.42
MAPK1 P28482 1/20 0.42
KCNA3 P22001 1/20 0.41
ADRB2 P07550 1/20 0.40
LMNA P02545 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
RXRA P19793 1/20 0.39
TSHR P16473 2/20 0.39
TP53 P04637 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5747450 0.96 HTR1B (0.52) HRH1SLC6A4HTR1BHTR1DHTR6
SCHEMBL5745853 0.88 HTR1B (0.53) HRH1SLC6A4HTR1BHTR6KDM4E
SCHEMBL5748300 0.88 HTR1B (0.56) HTR1BHTR1DHTR6KDM4EALDH1A1
SCHEMBL5747008 0.86 HTR1B (0.56) HTR1BHTR1DHTR6KDM4EALDH1A1
SCHEMBL5748074 0.85 SLC6A4 (0.53) HRH1SLC6A4HTR1BHTR1DHTR6
SCHEMBL5747032 0.85 HTR1B (0.49) HTR1BHTR6ALDH1A1KCNA3LMNA
SCHEMBL5749144 0.83 HTR1B (0.48) HTR1BHTR6KDM4EHPGDMAPK1
SCHEMBL5747914 0.81 HTR1B (0.52) HRH1SLC6A4HTR1BHTR1DHTR6
SCHEMBL5745052 0.81 SLC6A4 (0.46) HRH1SLC6A4HTR1BHTR1DKDM4E
SCHEMBL5748004 0.81 CYP2D6 (0.50) HTR6ALDH1A1TDP1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1711463-A2 AMINO-SUBSTITUTED TRICYCLIC DERIVATIVES AND METHODS OF USE ABBOTT LABORATORIES (US) 2006-10-18 EP claimed
WO-2005077899-A2 AMINO-SUBSTITUTED TRICYCLIC DERIVATIVES AND METHODS OF USE ABBOTT LABORATORIES (US) 2005-08-25 WO claimed