SCHEMBL5747008

SCHEMBL5747008

CCCNCCOc1cccc2c1c1ccccc1c(=O)n2C

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1B P28222 4/20 0.56
HEXA P06865 1/20 0.42
HEXB P07686 1/20 0.42
ADRB2 P07550 2/20 0.42
HTR1D P28221 2/20 0.41
KDM4E B2RXH2 3/20 0.39
ALDH1A1 P00352 3/20 0.39
MAPK1 P28482 2/20 0.39
HPGD P15428 2/20 0.39
HSD17B10 Q99714 2/20 0.39
HTR1A P08908 1/20 0.39
ADRA1D P25100 1/20 0.39
ADRA1A P35348 1/20 0.39
ADRA1B P35368 1/20 0.39
MEN1 O00255 1/20 0.38
USP2 O75604 1/20 0.38
LMNA P02545 1/20 0.38
HTT P42858 1/20 0.38
RECQL P46063 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5748300 0.91 HTR1B (0.56) HTR1BHEXAHEXBADRB2HTR1D
SCHEMBL5745853 0.89 HTR1B (0.53) HTR1BHEXAHEXBADRB2KDM4E
SCHEMBL5747450 0.88 HTR1B (0.52) HTR1BHEXAHEXBHTR1DKDM4E
SCHEMBL5750596 0.86 HRH1 (0.53) HTR1BADRB2HTR1DKDM4EALDH1A1
SCHEMBL5749144 0.82 HTR1B (0.48) HTR1BKDM4EMAPK1HPGDMEN1
SCHEMBL5747032 0.81 HTR1B (0.49) HTR1BALDH1A1LMNAHTTSMN1; SMN2
SCHEMBL5745160 0.81 HTR1B (0.46) HTR1BHTR1DKDM4EALDH1A1HPGD
SCHEMBL5745052 0.80 SLC6A4 (0.46) HTR1BHTR1DKDM4EALDH1A1HPGD
SCHEMBL5749009 0.79 HTR1B (0.56) HTR1BHEXAHEXBADRB2HTR1D
SCHEMBL5771872 0.79 HTR1B (0.60) HTR1BHEXAHEXBADRB2HTR1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1711463-A2 AMINO-SUBSTITUTED TRICYCLIC DERIVATIVES AND METHODS OF USE ABBOTT LABORATORIES (US) 2006-10-18 EP claimed
WO-2005077899-A2 AMINO-SUBSTITUTED TRICYCLIC DERIVATIVES AND METHODS OF USE ABBOTT LABORATORIES (US) 2005-08-25 WO claimed