SCHEMBL5751074

SCHEMBL5751074

COc1ccc2nccc(NC(=O)OC3(O)CCN(CC(=O)c4ccc5c(c4)NC(=O)CS5)CC3)c2n1

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
HPGD P15428 1/20 0.40
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
KCNH2 Q12809 2/20 0.37
POLB P06746 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6667019 0.90 KCNH2 (0.45) NPC1RAB9AALDH1A1LMNAHPGD
SCHEMBL5750711 0.88 KCNH2 (0.40) MEN1KMT2AKCNH2
SCHEMBL5765739 0.88 ALDH1A1 (0.40) NPC1RAB9AALDH1A1LMNAHPGD
SCHEMBL14573152 0.86 KCNH2 (0.44) NPC1RAB9AALDH1A1LMNAHPGD
SCHEMBL5748821 0.84 KCNH2 (0.39) HPGDMEN1KMT2AKCNH2
SCHEMBL5751255 0.81 KCNH2 (0.38) MEN1KMT2AKCNH2
SCHEMBL5750809 0.80 KCNH2 (0.38) MEN1KMT2AKCNH2
SCHEMBL5749450 0.80 KCNH2 (0.39) KCNH2
SCHEMBL5747711 0.80 KCNH2 (0.38) MEN1KMT2AKCNH2POLB
SCHEMBL5656474 0.80 HTR1A (0.47) ALDH1A1LMNAHPGDKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1419155-B1 PIPERIDINE DERIVATIVES AS ANTIBACTERIAL AGENTS SMITHKLINE BEECHAM PLC (GB) 2006-11-08 EP claimed