SCHEMBL5765739

SCHEMBL5765739

COc1ccc2nccc(NC(=O)OC3CCN(CC(=O)c4ccc5c(c4)NC(=O)CS5)CC3)c2n1

nearest known ligand 0.51

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
KCNH2 Q12809 3/20 0.40
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
HPGD P15428 1/20 0.39
HTR1D P28221 2/20 0.38
HTR1A P08908 1/20 0.38
HTR1B P28222 1/20 0.38
EIF4H Q15056 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14573152 0.90 KCNH2 (0.44) ALDH1A1LMNAKCNH2NPC1RAB9A
SCHEMBL5751074 0.88 NPC1 (0.41) ALDH1A1LMNAKCNH2NPC1RAB9A
SCHEMBL5764669 0.88 KCNH2 (0.45) KCNH2
SCHEMBL5767030 0.86 SLC2A1 (0.43) KCNH2
SCHEMBL5764977 0.86 HTR1D (0.53) ALDH1A1KCNH2HTR1DHTR1AHTR1B
SCHEMBL6667019 0.86 KCNH2 (0.45) ALDH1A1LMNAKCNH2NPC1RAB9A
SCHEMBL5656474 0.84 HTR1A (0.47) ALDH1A1LMNAKCNH2HPGDHTR1D
SCHEMBL5762645 0.81 KCNH2 (0.53) ALDH1A1LMNAKCNH2NPC1RAB9A
SCHEMBL5765126 0.80 SLC2A1 (0.43) KCNH2
SCHEMBL14573142 0.78 KCNH2 (0.44) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1392686-B1 BICYCLIC NITROGEN-CONTAINING HETEROCYCLIC DERIVATIVES FOR USE AS ANTIBACTERIALS SMITHKLINE BEECHAM PLC (GB) 2006-10-18 EP claimed