SCHEMBL5754433

SCHEMBL5754433

C=CC(CN1CCN(Cc2ccccc2)CC1)Oc1ccc(F)cc1

nearest known ligand 0.53

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.53
HTT P42858 1/20 0.53
CACNA1G O43497 3/20 0.47
SIGMAR1 Q99720 3/20 0.46
KCNH2 Q12809 1/20 0.46
SLC6A3 Q01959 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5752956 0.79 KDM4E (0.54) KDM4EHTTCACNA1GSIGMAR1KCNH2
SCHEMBL10362355 0.77 KDM4E (0.74) KDM4EHTTSIGMAR1SLC6A3
Hydrochloric Acid SCHEMBL7299429 0.76 KDM4E (0.76) KDM4EHTTSIGMAR1SLC6A3
SCHEMBL8725812 0.74 SIGMAR1 (0.75) KDM4EHTTSIGMAR1
SCHEMBL7423189 0.71 SIGMAR1 (0.69) KDM4EHTTSIGMAR1
SCHEMBL8029920 0.70 LTA4H (0.65) KDM4EHTTSIGMAR1
SCHEMBL8035741 0.69 ALDH1A1 (0.54)
SCHEMBL8035719 0.69 LTA4H (0.63) KDM4ECACNA1GSIGMAR1KCNH2
SCHEMBL8238268 0.68 SLC6A2 (0.40) KDM4EHTTCACNA1GSIGMAR1KCNH2
SCHEMBL16226160 0.68 KDM4E (0.72) KDM4EHTTSIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1099692-B1 N,N-SUBSTITUTED CYCLIC AMINE DERIVATIVES EISAI CO LTD (JP) 2006-05-03 EP disclosed
US-6737425-B1 SUCH AS 1-((4-CYANO-5-METHYL-4-PHENYL)HEXYL)-4-(2-(4-FLUORO -PHENOXY)ETHYL)PIPERAZINE; NERVE SELECTIVE CALCIUM ANTAGONISTS EISAI CO., LTD. (JP) 2004-05-18 US disclosed
EP-1099692-A1 N,N-SUBSTITUTED CYCLIC AMINE DERIVATIVES Eisai Co., Ltd. (JP) 2001-05-16 EP disclosed