SCHEMBL5754473

SCHEMBL5754473

CC(C)C(C#N)(CCCN1CCN(CCO)CC1)c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.49
EBP Q15125 2/20 0.49
CCR3 P51677 2/20 0.49
CHRM4 P08173 4/20 0.48
CHRM3 P20309 4/20 0.48
CHRM5 P08912 3/20 0.48
CHRM2 P08172 2/20 0.47
CHRM1 P11229 2/20 0.47
CCR1 P32246 3/20 0.46
RAB9A P51151 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
CACNA1B Q00975 2/20 0.46
KDM4E B2RXH2 1/20 0.43
HTR1A P08908 1/20 0.43
CYP2D6 P10635 1/20 0.43
DRD2 P14416 1/20 0.43
DRD1 P21728 1/20 0.43
HTR2A P28223 1/20 0.43
OPRM1 P35372 1/20 0.43
DRD3 P35462 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14431859 0.94 CCR3 (0.54) SIGMAR1EBPCCR3CHRM4CHRM3
SCHEMBL5240018 0.91 RAB9A (0.52) SIGMAR1EBPCCR3CHRM4CHRM3
SCHEMBL14431920 0.90 RAB9A (0.58) SIGMAR1EBPCCR3CHRM4CHRM3
SCHEMBL14431854 0.90 SIGMAR1 (0.51) SIGMAR1EBPCCR3CHRM4CHRM3
SCHEMBL5750440 0.88 CCR3 (0.52) SIGMAR1EBPCCR3CHRM4CHRM3
SCHEMBL5237846 0.86 SIGMAR1 (0.60) SIGMAR1EBPCCR3CHRM4CHRM3
SCHEMBL5239804 0.86 KCNA3 (0.60) SIGMAR1EBPCCR3CHRM4CHRM3
SCHEMBL5239794 0.86 SIGMAR1 (0.60) SIGMAR1EBPCCR3KCNA3
SCHEMBL14431875 0.86 CCR3 (0.49) SIGMAR1EBPCCR3CHRM4CHRM3
SCHEMBL5235995 0.86 CHRM4 (0.54) SIGMAR1EBPCCR3CHRM4CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1099692-B1 N,N-SUBSTITUTED CYCLIC AMINE DERIVATIVES EISAI CO LTD (JP) 2006-05-03 EP disclosed
US-6737425-B1 SUCH AS 1-((4-CYANO-5-METHYL-4-PHENYL)HEXYL)-4-(2-(4-FLUORO -PHENOXY)ETHYL)PIPERAZINE; NERVE SELECTIVE CALCIUM ANTAGONISTS EISAI CO., LTD. (JP) 2004-05-18 US disclosed
EP-1099692-A1 N,N-SUBSTITUTED CYCLIC AMINE DERIVATIVES Eisai Co., Ltd. (JP) 2001-05-16 EP disclosed