SCHEMBL5754907

SCHEMBL5754907

Fc1ccc(CCCN2CCNCC2)cc1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 9/20 0.70
KCNH2 Q12809 3/20 0.59
SLC6A2 P23975 2/20 0.59
SLC6A4 P31645 2/20 0.59
SLC6A3 Q01959 2/20 0.59
SCN5A Q14524 1/20 0.54
DRD2 P14416 3/20 0.51
HTR1A P08908 2/20 0.51
DRD1 P21728 2/20 0.51
DRD5 P21918 2/20 0.51
HTR2A P28223 2/20 0.51
DRD3 P35462 2/20 0.51
TMEM97 Q5BJF2 1/20 0.51
MEN1 O00255 1/20 0.49
NPC1 O15118 1/20 0.49
ALDH1A1 P00352 1/20 0.49
LMNA P02545 1/20 0.49
TP53 P04637 1/20 0.49
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10507686 0.95 SIGMAR1 (0.63) SIGMAR1KCNH2SLC6A2SLC6A4SLC6A3
SCHEMBL2549429 0.89 KCNH2 (0.71) SIGMAR1KCNH2SLC6A2SLC6A4SLC6A3
Hydrochloric Acid SCHEMBL5410232 0.88 KCNH2 (0.69) SIGMAR1KCNH2SLC6A2SLC6A4SLC6A3
Hydrochloric Acid SCHEMBL2548737 0.88 KCNH2 (0.69) SIGMAR1KCNH2SLC6A2SLC6A4SLC6A3
SCHEMBL22813547 0.84 SCN5A (0.71) SIGMAR1SLC6A4SLC6A3SCN5ADRD2
SCHEMBL5752571 0.83 KCNH2 (0.64) SIGMAR1KCNH2SLC6A2SLC6A4SLC6A3
SCHEMBL11630606 0.83 SIGMAR1 (0.70) SIGMAR1KCNH2SLC6A4MEN1NPC1
SCHEMBL15651128 0.83 SIGMAR1 (0.70) SIGMAR1KCNH2SLC6A2SLC6A4SLC6A3
SCHEMBL9319743 0.83 SIGMAR1 (0.70) SIGMAR1KCNH2SLC6A2SLC6A4SLC6A3
SCHEMBL13858201 0.83 SIGMAR1 (0.70) SIGMAR1KCNH2SLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1099692-B1 N,N-SUBSTITUTED CYCLIC AMINE DERIVATIVES EISAI CO LTD (JP) 2006-05-03 EP disclosed
US-6737425-B1 SUCH AS 1-((4-CYANO-5-METHYL-4-PHENYL)HEXYL)-4-(2-(4-FLUORO -PHENOXY)ETHYL)PIPERAZINE; NERVE SELECTIVE CALCIUM ANTAGONISTS EISAI CO., LTD. (JP) 2004-05-18 US disclosed
EP-1099692-A1 N,N-SUBSTITUTED CYCLIC AMINE DERIVATIVES Eisai Co., Ltd. (JP) 2001-05-16 EP disclosed