SCHEMBL5752571

SCHEMBL5752571

Fc1ccc(CCN2CCCNCC2)cc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 0.64
SLC6A4 P31645 2/20 0.64
SLC6A2 P23975 1/20 0.64
SLC6A3 Q01959 1/20 0.64
SIGMAR1 Q99720 4/20 0.62
CXCR4 P61073 5/20 0.54
HRH3 Q9Y5N1 2/20 0.54
MEN1 O00255 1/20 0.54
CHRM2 P08172 1/20 0.54
CHRM1 P11229 1/20 0.54
ADRA2C P18825 1/20 0.54
CCR2 P41597 1/20 0.54
CXCL12 P48061 1/20 0.54
BLM P54132 1/20 0.54
KMT2A Q03164 1/20 0.54
TDP1 Q9NUW8 1/20 0.54
KCNJ1 P48048 2/20 0.54
MAOA P21397 1/20 0.50
MBTD1 Q05BQ5 1/20 0.50
L3MBTL3 Q96JM7 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2549429 0.93 KCNH2 (0.71) KCNH2SLC6A4SLC6A2SLC6A3SIGMAR1
Hydrochloric Acid SCHEMBL5410232 0.92 KCNH2 (0.69) KCNH2SLC6A4SLC6A2SLC6A3SIGMAR1
Hydrochloric Acid SCHEMBL2548737 0.92 KCNH2 (0.69) KCNH2SLC6A4SLC6A2SLC6A3SIGMAR1
SCHEMBL23377845 0.84 HRH3 (0.62) KCNH2SLC6A3SIGMAR1HRH3TDP1
SCHEMBL23377646 0.84 HRH3 (0.68) KCNH2SLC6A3SIGMAR1HRH3TDP1
SCHEMBL22254774 0.84 HRH3 (0.72) KCNH2SLC6A4SLC6A2SLC6A3SIGMAR1
SCHEMBL2003768 0.83 CXCR4 (0.77) SIGMAR1CXCR4HRH3MEN1CHRM2
SCHEMBL8668531 0.83 SLC6A3 (0.70) KCNH2SLC6A4SLC6A3SIGMAR1CXCR4
SCHEMBL5754907 0.83 SIGMAR1 (0.70) KCNH2SLC6A4SLC6A2SLC6A3SIGMAR1
SCHEMBL9397186 0.83 SIGMAR1 (0.58) KCNH2SLC6A4SLC6A2SLC6A3SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1099692-B1 N,N-SUBSTITUTED CYCLIC AMINE DERIVATIVES EISAI CO LTD (JP) 2006-05-03 EP disclosed
US-6737425-B1 SUCH AS 1-((4-CYANO-5-METHYL-4-PHENYL)HEXYL)-4-(2-(4-FLUORO -PHENOXY)ETHYL)PIPERAZINE; NERVE SELECTIVE CALCIUM ANTAGONISTS EISAI CO., LTD. (JP) 2004-05-18 US disclosed
EP-1099692-A1 N,N-SUBSTITUTED CYCLIC AMINE DERIVATIVES Eisai Co., Ltd. (JP) 2001-05-16 EP disclosed