SCHEMBL5755250

SCHEMBL5755250

CC(=O)OOc1ccc(F)cc1OC(C)=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.46
ALDH1A1 P00352 4/20 0.46
TSHR P16473 3/20 0.46
GAA P10253 2/20 0.46
RAB9A P51151 1/20 0.46
CYP4F2 P78329 1/20 0.41
CYP4A11 Q02928 1/20 0.41
CFD P00746 2/20 0.41
AMY1A P0DUB6 1/20 0.40
BLM P54132 2/20 0.40
TDP1 Q9NUW8 2/20 0.40
HPGD P15428 2/20 0.40
HSD17B10 Q99714 2/20 0.40
TNFSF11 O14788 1/20 0.40
ESR1 P03372 1/20 0.40
ITGB3 P05106 1/20 0.40
ITGA2B P08514 1/20 0.40
HMGB1 P09429 1/20 0.40
GGT1 P19440 1/20 0.40
PTGS1 P23219 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5755257 0.87 TSHR (0.58) KDM4EALDH1A1TSHRGAARAB9A
SCHEMBL5740669 0.82 CES2 (0.42) RAB9AHPGDMAPTKMT2AL3MBTL1
SCHEMBL27674522 0.81 CA3 (0.41) GAACA9CYP2C19
SCHEMBL6649289 0.81 FFAR1 (0.44) KDM4EALDH1A1TSHRRAB9AHPGD
SCHEMBL27692981 0.79 NPC1 (0.42) KDM4EALDH1A1RAB9AHPGDPOLB
SCHEMBL5756842 0.79 ALDH1A1 (0.44) ALDH1A1TSHRGAAKMT2A
SCHEMBL2908009 0.79 TSHR (0.62) KDM4EALDH1A1TSHRGAARAB9A
SCHEMBL823700 0.78 CYP4F2 (0.50) KDM4EALDH1A1TSHRGAARAB9A
SCHEMBL1991907 0.78 CYP4F2 (0.64) KDM4EALDH1A1TSHRGAARAB9A
SCHEMBL11355453 0.78 ALDH1A1 (0.40) KDM4EALDH1A1GAAMAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1099692-B1 N,N-SUBSTITUTED CYCLIC AMINE DERIVATIVES EISAI CO LTD (JP) 2006-05-03 EP disclosed
US-6737425-B1 SUCH AS 1-((4-CYANO-5-METHYL-4-PHENYL)HEXYL)-4-(2-(4-FLUORO -PHENOXY)ETHYL)PIPERAZINE; NERVE SELECTIVE CALCIUM ANTAGONISTS EISAI CO., LTD. (JP) 2004-05-18 US disclosed
EP-1099692-A1 N,N-SUBSTITUTED CYCLIC AMINE DERIVATIVES Eisai Co., Ltd. (JP) 2001-05-16 EP disclosed