SCHEMBL5756154

SCHEMBL5756154

Cc1ccc(C(=O)N(CCCNC(=O)OC(C)(C)C)CC(C)Cc2nc(C)c(C#N)c(=O)n2Cc2ccccc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 12/20 0.51
KCNH2 Q12809 2/20 0.38
FNTA P49354 1/20 0.38
FNTB P49356 1/20 0.38
PGGT1B P53609 1/20 0.38
CYP3A4 P08684 2/20 0.37
CYP2C19 P33261 2/20 0.37
ALDH1A1 P00352 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
MC4R P32245 1/20 0.37
KIF23 Q02241 1/20 0.36
CTSS P25774 2/20 0.35
CTSL P07711 1/20 0.35
CTSB P07858 1/20 0.35
CTSK P43235 1/20 0.35
MAP1LC3B Q9GZQ8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5247152 0.86 KIF11 (0.52) KIF11KCNH2CYP3A4CYP2C19MC4R
SCHEMBL5248554 0.86 KIF11 (0.49) KIF11KCNH2CYP3A4CYP2C19MC4R
SCHEMBL5756151 0.82 KIF11 (0.60) KIF11KCNH2CYP3A4CYP2C19KIF23
SCHEMBL4363439 0.77 KIF11 (0.58) KIF11
SCHEMBL4376313 0.76 KIF11 (0.57) KIF11
SCHEMBL4366741 0.75 KIF11 (0.54) KIF11KCNH2CYP3A4CYP2C19KIF23
SCHEMBL3905973 0.75 KIF11 (0.51) KIF11MC4RKIF23GNRHR
SCHEMBL5246236 0.75 KIF11 (0.52) KIF11MC4RKIF23GNRHR
SCHEMBL5756255 0.74 KIF11 (0.51) KIF11KCNH2CYP3A4CYP2C19ALDH1A1
SCHEMBL13956801 0.74 KIF11 (0.64) KIF11KCNH2CYP3A4CYP2C19KIF23

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1503993-A4 COMPOUNDS, METHODS AND COMPOSITIONS CYTOKINETICS INC (US) 2006-05-03 EP disclosed
EP-1503993-A2 COMPOUNDS, METHODS AND COMPOSITIONS Cytokinetics, Inc. (US) 2005-02-09 EP disclosed
WO-2003094839-A2 PYRIMIDINONE COMPOUNDS, COMPOSITIONS AND METHODS CYTOKINETICS, INC. (US) 2003-11-20 WO disclosed