SCHEMBL5756300

SCHEMBL5756300

Cc1ccc(-n2cc(CNC(=O)c3ccc(C)n(-c4cccc(C(F)(F)F)c4)c3=O)cn2)cc1

nearest known ligand 0.63

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ELANE P08246 4/20 0.63
CCR1 P32246 13/20 0.48
DDT P30046 2/20 0.48
MAPK1 P28482 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5757939 0.95 ELANE (0.65) ELANECCR1DDT
SCHEMBL27643790 0.93 ELANE (0.64) ELANECCR1DDT
SCHEMBL5757082 0.93 ELANE (0.63) ELANECCR1DDT
SCHEMBL27624435 0.89 ELANE (0.61) ELANECCR1DDT
SCHEMBL5757244 0.88 ELANE (0.67) ELANECCR1DDTMAPK1
SCHEMBL5758770 0.87 ELANE (0.80) ELANECCR1DDTNPSR1
SCHEMBL5757669 0.86 ELANE (0.65) ELANECCR1DDT
SCHEMBL5757950 0.83 ELANE (0.69) ELANECCR1DDT
SCHEMBL5758687 0.82 ELANE (0.73) ELANECCR1DDT
SCHEMBL5755788 0.82 ELANE (0.79) ELANECCR1DDT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1562902-B1 2-PYRIDONE DERIVATIVES AS INHIBITORS OF NEUTROPHILE ELASTASE ASTRAZENECA AB (SE) 2006-05-03 EP disclosed
US-20060035938-A1 2-Pyridone derivatives as inhibitors of neutrophile elastase ASRAZENECA AB (SE) 2006-02-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060035938-A1 2-Pyridone derivatives as inhibitors of neutrophile elastase SERPINB1, ELANE, SERPINE1 ELANE 2/4885CCR1 186/4885DDT 3860/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.