SCHEMBL5757082

SCHEMBL5757082

Cc1cccc(-n2cc(CNC(=O)c3ccc(C)n(-c4cccc(C(F)(F)F)c4)c3=O)cn2)c1

nearest known ligand 0.63

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ELANE P08246 4/20 0.63
DDT P30046 2/20 0.54
CCR1 P32246 10/20 0.46
EPHX2 P34913 1/20 0.43
NPY5R Q15761 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5756300 0.93 ELANE (0.63) ELANEDDTCCR1
SCHEMBL5757939 0.93 ELANE (0.65) ELANEDDTCCR1EPHX2
SCHEMBL27624435 0.91 ELANE (0.61) ELANEDDTCCR1EPHX2
SCHEMBL27643790 0.90 ELANE (0.64) ELANEDDTCCR1
SCHEMBL5757244 0.88 ELANE (0.67) ELANEDDTCCR1
SCHEMBL5440126 0.87 DDT (0.51) ELANEDDTCCR1
SCHEMBL5758687 0.86 ELANE (0.73) ELANEDDTCCR1
SCHEMBL5757669 0.86 ELANE (0.65) ELANEDDTCCR1
SCHEMBL5758770 0.83 ELANE (0.80) ELANEDDTCCR1
SCHEMBL5755788 0.82 ELANE (0.79) ELANEDDTCCR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1562902-B1 2-PYRIDONE DERIVATIVES AS INHIBITORS OF NEUTROPHILE ELASTASE ASTRAZENECA AB (SE) 2006-05-03 EP disclosed
US-20060035938-A1 2-Pyridone derivatives as inhibitors of neutrophile elastase ASRAZENECA AB (SE) 2006-02-16 US disclosed
EP-1562902-A1 2-PYRIDONE DERIVATIVES AS INHIBITORS OF NEUTROPHILE ELASTASE AstraZeneca AB (SE) 2005-08-17 EP disclosed
WO-2004043924-A1 2-PYRIDONE DERIVATIVES AS INHIBITORS OF NEUTROPHILE ELASTASE ASTRAZENECA AB (SE) 2004-05-27 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060035938-A1 2-Pyridone derivatives as inhibitors of neutrophile elastase SERPINB1, ELANE, SERPINE1 ELANE 2/4885DDT 3860/4885CCR1 186/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.