SCHEMBL5756520

SCHEMBL5756520

CN(C)CCN(C)C(=O)c1ccc2nc(-c3c(O)cccc3OCc3ccc(C(=O)O)cc3)sc2c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.41
KDM4E B2RXH2 2/20 0.41
NFKB1 P19838 2/20 0.41
NFKB2 Q00653 2/20 0.41
RELA Q04206 2/20 0.41
LMNA P02545 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
NPC1 O15118 3/20 0.41
RAB9A P51151 2/20 0.41
LTB4R Q15722 1/20 0.40
LTB4R2 Q9NPC1 1/20 0.40
RXRA P19793 3/20 0.39
RXRB P28702 2/20 0.39
RXRG P48443 2/20 0.39
ILK Q13418 1/20 0.37
MITF O75030 1/20 0.37
ALDH1A1 P00352 1/20 0.37
POLB P06746 1/20 0.37
GAA P10253 1/20 0.37
MAPT P10636 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5761323 0.93 CYP3A4 (0.45) EGFRKDM4ELMNASMN1; SMN2NPC1
SCHEMBL5756078 0.74 KDM4E (0.55) KDM4ENFKB1NFKB2RELALMNA
SCHEMBL5757301 0.72 KDM4E (0.48) KDM4ENFKB1NFKB2RELALMNA
SCHEMBL5757292 0.71 KMT2A (0.48) LMNASMN1; SMN2NPC1RAB9AALDH1A1
SCHEMBL5758746 0.71 MGAM (0.47) KDM4ELMNASMN1; SMN2NPC1RAB9A
SCHEMBL5756311 0.70 ROCK2 (0.45) NFKB1NFKB2RELASMN1; SMN2NPC1
SCHEMBL5755215 0.64 MAPK1 (0.52) KDM4ELMNASMN1; SMN2NPC1RAB9A
SCHEMBL5757590 0.64 CA2 (0.52) KDM4ESMN1; SMN2NPC1RAB9AALDH1A1
SCHEMBL5759668 0.64 KDM4E (0.51) KDM4ENFKB1NFKB2RELALMNA
SCHEMBL6104213 0.63 GAA (0.44) KDM4ENFKB1NFKB2RELALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539723-B1 NOVEL USE OF BENZOTHIAZOLE DERIVATIVES ASTRAZENECA AB (SE) 2006-05-24 EP claimed