SCHEMBL5756778

SCHEMBL5756778

COc1ccc(CC(SCC2CCCCC2)C(CNC(=O)c2ccccc2O)NC(=O)[C@@H]2CSCN2C(=O)OC(C)(C)C)cc1OCc1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 1/20 0.38
HSD17B10 Q99714 1/20 0.36
ATM Q13315 1/20 0.35
NPC1 O15118 3/20 0.35
RAB9A P51151 2/20 0.35
PKM P14618 1/20 0.35
YAP1 P46937 3/20 0.34
CTSD P07339 2/20 0.33
GHSR Q92847 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
HDAC3 O15379 1/20 0.33
HDAC4 P56524 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC7 Q8WUI4 1/20 0.33
HDAC2 Q92769 1/20 0.33
HDAC10 Q969S8 1/20 0.33
HDAC11 Q96DB2 1/20 0.33
HDAC8 Q9BY41 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5758199 0.91 CACNA1B (0.43) CACNA1BHSD17B10ATMYAP1GHSR
SCHEMBL5754912 0.88 CACNA1B (0.43) CACNA1BHSD17B10ATMYAP1MEN1
SCHEMBL5758645 0.88 CACNA1B (0.43) CACNA1BHSD17B10ATMYAP1MEN1
SCHEMBL5754050 0.87 NPC1 (0.37) CACNA1BNPC1RAB9APKMCTSD
SCHEMBL5759035 0.86 CACNA1B (0.49) CACNA1BHSD17B10ATMYAP1GHSR
SCHEMBL5754736 0.85 CACNA1B (0.40) CACNA1BHSD17B10ATMMEN1KMT2A
SCHEMBL5753816 0.85 NPC1 (0.37) NPC1RAB9APKMCTSDMEN1
SCHEMBL5756658 0.84 CACNA1B (0.39) CACNA1BHSD17B10ATMMEN1KMT2A
SCHEMBL5757036 0.83 CACNA1B (0.45) CACNA1BHSD17B10KMT2A
SCHEMBL5755981 0.82 KMT2A (0.38) CACNA1BHSD17B10YAP1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0997147-B1 AMINO ACID DERIVATIVES ONO PHARMACEUTICAL CO (JP) 2006-03-15 EP claimed