SCHEMBL5757186

SCHEMBL5757186

CC(Cl)c1cc(F)ccc1S(=O)(=O)c1ccc(F)cc1C(C)Cl

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PSEN1 P49768 6/20 0.47
PSEN2 P49810 6/20 0.47
APH1B Q8WW43 6/20 0.47
NCSTN Q92542 6/20 0.47
APH1A Q96BI3 6/20 0.47
PSENEN Q9NZ42 6/20 0.47
HTR2A P28223 2/20 0.36
HTR2C P28335 2/20 0.36
KCNH2 Q12809 2/20 0.36
AKR1B1 P15121 2/20 0.35
KMT2A Q03164 1/20 0.35
PTGES2 Q9H7Z7 1/20 0.35
KDM4E B2RXH2 1/20 0.34
CCR2 P41597 1/20 0.34
CNR1 P21554 1/20 0.33
TRPV4 Q9HBA0 1/20 0.33
RXFP1 Q9HBX9 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5957556 0.79 TRPV4 (0.41) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL2814293 0.74 PSEN1 (0.44) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL587387 0.72 MMP2 (0.44) HTR2AHTR2CKCNH2KMT2AKDM4E
SCHEMBL18929871 0.72 PSEN1 (0.41) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL20817934 0.71 PSEN1 (0.37) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL31574267 0.71 PSEN1 (0.37) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL13797487 0.70 AKR1B1 (0.44) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL896792 0.70 TSHR (0.50) AKR1B1KMT2ARXFP1
SCHEMBL2122256 0.70 TSHR (0.50) AKR1B1KMT2ARXFP1
SCHEMBL9963191 0.69 POLB (0.45) PSEN1PSEN2APH1BNCSTNAPH1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1099692-B1 N,N-SUBSTITUTED CYCLIC AMINE DERIVATIVES EISAI CO LTD (JP) 2006-05-03 EP disclosed
US-6737425-B1 SUCH AS 1-((4-CYANO-5-METHYL-4-PHENYL)HEXYL)-4-(2-(4-FLUORO -PHENOXY)ETHYL)PIPERAZINE; NERVE SELECTIVE CALCIUM ANTAGONISTS EISAI CO., LTD. (JP) 2004-05-18 US disclosed