SCHEMBL5757459

SCHEMBL5757459

CS(=O)(=O)c1ccc(CBr)cc1Cl.CS(=O)(=O)c1ccc(CO)cc1Cl

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1D P25100 1/20 0.43
CYP4F2 P78329 1/20 0.39
CYP4A11 Q02928 1/20 0.39
PTGDR2 Q9Y5Y4 1/20 0.38
PTGES2 Q9H7Z7 2/20 0.35
CCR2 P41597 1/20 0.35
NPC1 O15118 1/20 0.35
HPGD P15428 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.34
PTGS2 P35354 1/20 0.34
PIK3CD O00329 1/20 0.34
PIK3CA P42336 1/20 0.34
PIK3CB P42338 1/20 0.34
PIK3CG P48736 1/20 0.34
NR1H2 P55055 1/20 0.33
NR1H3 Q13133 1/20 0.33
CMA1 P23946 1/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29595036 0.92 ADRA1D (0.44) ADRA1DCYP4F2CYP4A11PTGDR2CCR2
SCHEMBL6196958 0.92 ADRA1D (0.47) ADRA1DPTGDR2PTGES2CCR2NPC1
SCHEMBL1013697 0.92 ADRA1D (0.44) ADRA1DCYP4F2CYP4A11PTGDR2CCR2
SCHEMBL5756525 0.83 CA2 (0.37) PTGES2RAB9AL3MBTL1PTGS2PIK3CD
SCHEMBL5760478 0.81 ADRA1D (0.40) ADRA1DPTGDR2PTGES2CCR2NPC1
SCHEMBL27624382 0.79 ADRA1D (0.42) ADRA1DPTGDR2PTGES2CCR2L3MBTL1
SCHEMBL1013610 0.78 GSTO1 (0.44) PTGES2CCR2SMN1; SMN2L3MBTL1PTGS2
SCHEMBL1015882 0.78 GSTO1 (0.44) CYP4F2CYP4A11CCR2HPGDSMN1; SMN2
Hydrochloric Acid SCHEMBL27763840 0.77 CYP4F2 (0.40) ADRA1DCYP4F2CYP4A11PTGES2HPGD
SCHEMBL13211313 0.76 ADRA1D (0.45) ADRA1DPTGDR2CCR2NPC1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611088-A2 HYDROXAMATES AS THERAPEUTIC AGENTS AXYS PHARMACEUTICALS, INC. (US) 2006-01-04 EP claimed
WO-2004092115-A2 HYDROXAMATES AS THERAPEUTIC AGENTS AXYS PHARMACEUTICALS INC. (US) 2004-10-28 WO claimed