SCHEMBL5757544

SCHEMBL5757544

COc1ccc(-c2n[nH]cc2Cc2ccncc2)cc1OC1CCCO1

nearest known ligand 0.41

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 10/20 0.41
PDE4B Q07343 6/20 0.40
S1PR1 P21453 2/20 0.39
S1PR3 Q99500 1/20 0.39
CYP17A1 P05093 1/20 0.37
PDE4D Q08499 5/20 0.37
PDE4C Q08493 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5755717 0.91 PDE4B (0.44) PDE4APDE4BPDE4DPDE4C
SCHEMBL5755076 0.86 PDE4B (0.44) PDE4APDE4BPDE4DPDE4C
SCHEMBL5759793 0.84 PDE4A (0.41) PDE4APDE4BPDE4DPDE4C
SCHEMBL5759164 0.84 PDE4B (0.43) PDE4APDE4BPDE4DPDE4C
SCHEMBL5756380 0.82 PDE4B (0.41) PDE4APDE4BS1PR1S1PR3PDE4D
SCHEMBL5758859 0.82 PDE4B (0.41) PDE4APDE4BPDE4DPDE4C
SCHEMBL5758807 0.79 PDE4B (0.42) PDE4APDE4BS1PR1S1PR3PDE4D
SCHEMBL5756557 0.78 DHFR (0.33) PDE4APDE4BPDE4DPDE4C
SCHEMBL5759401 0.78 PDE4B (0.43) PDE4APDE4BPDE4DPDE4C
SCHEMBL5755003 0.76 PDE4B (0.42) PDE4APDE4BPDE4DPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1631568-A1 PYRAZOLE DERIVATIVES AS PHOSPHODIESTERASE 4 INHIBITORS Memory Pharmaceuticals Corporation (US) 2006-03-08 EP disclosed
WO-2004094411-A1 PYRAZOLE DERIVATIVES AS PHOSPHODIESTERASE 4 INHIBITORS MEMORY PHARMACEUTICALS CORPORATION (US) 2004-11-04 WO disclosed