SCHEMBL5759739

SCHEMBL5759739

Cc1cccc(-n2cccc(C(=O)O)c2=O)c1

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 2/20 0.52
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
ALKBH5 Q6P6C2 1/20 0.47
POLB P06746 2/20 0.45
ALDH1A1 P00352 6/20 0.44
PKM P14618 2/20 0.44
MAPT P10636 1/20 0.44
KDM4E B2RXH2 2/20 0.43
GAA P10253 1/20 0.43
HSP90AA1 P07900 1/20 0.42
MGLL Q99685 1/20 0.42
HPGD P15428 2/20 0.42
L3MBTL1 Q9Y468 1/20 0.41
PARP1 P09874 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26601369 0.83 AKR1C3 (0.49) NOTUMPOLBALDH1A1PKMMAPT
SCHEMBL9292198 0.82 HSP90AA1 (0.49) NOTUMMEN1KMT2AALKBH5ALDH1A1
SCHEMBL1137068 0.82 KDM4E (0.54) NOTUMMEN1KMT2APOLBALDH1A1
SCHEMBL4137779 0.78 NOTUM (0.53) NOTUMMEN1KMT2AALKBH5POLB
SCHEMBL4313192 0.78 ALDH1A1 (0.42) NOTUMMEN1KMT2APOLBALDH1A1
SCHEMBL1259232 0.76 ALDH1A1 (0.49) NOTUMMEN1KMT2APOLBALDH1A1
SCHEMBL4430908 0.76 ALDH1A1 (0.51) MEN1KMT2APOLBALDH1A1MAPT
SCHEMBL1260210 0.76 NOTUM (0.64) NOTUMMEN1KMT2AALKBH5POLB
SCHEMBL2676151 0.75 KDM4E (0.73) NOTUMMEN1KMT2AALDH1A1KDM4E
SCHEMBL25529181 0.75 KDM4E (0.40) MEN1KMT2APOLBALDH1A1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1562902-B1 2-PYRIDONE DERIVATIVES AS INHIBITORS OF NEUTROPHILE ELASTASE ASTRAZENECA AB (SE) 2006-05-03 EP disclosed
US-20060035938-A1 2-Pyridone derivatives as inhibitors of neutrophile elastase ASRAZENECA AB (SE) 2006-02-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060035938-A1 2-Pyridone derivatives as inhibitors of neutrophile elastase SERPINB1, ELANE, SERPINE1 NOTUM 3748/4885MEN1 3423/4885KMT2A 4487/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.