SCHEMBL4313192

SCHEMBL4313192

Cc1ccc(C)c(-n2cccc(C(=O)O)c2=O)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.42
POLB P06746 3/20 0.42
TDP1 Q9NUW8 2/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
APEX1 P27695 1/20 0.42
HSD17B10 Q99714 1/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
SIRT5 Q9NXA8 1/20 0.41
AKR1C3 P42330 1/20 0.41
CSNK2A1 P68400 1/20 0.40
MPI P34949 2/20 0.40
PHOSPHO1 Q8TCT1 2/20 0.40
PMM2 O15305 1/20 0.40
KDM4E B2RXH2 1/20 0.40
GAA P10253 1/20 0.40
PKM P14618 1/20 0.40
NOTUM Q6P988 1/20 0.39
NSD2 O96028 1/20 0.39
MAPT P10636 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1260115 0.83 POLB (0.53) ALDH1A1POLBTDP1L3MBTL1APEX1
SCHEMBL26601369 0.78 AKR1C3 (0.49) ALDH1A1POLBTDP1L3MBTL1APEX1
SCHEMBL5759739 0.78 NOTUM (0.52) ALDH1A1POLBL3MBTL1MEN1KMT2A
SCHEMBL1260315 0.77 P2RX7 (0.42) ALDH1A1POLBTDP1L3MBTL1APEX1
SCHEMBL4628972 0.75 POLB (0.63) ALDH1A1POLBTDP1L3MBTL1APEX1
SCHEMBL1259232 0.75 ALDH1A1 (0.49) ALDH1A1POLBTDP1L3MBTL1APEX1
SCHEMBL5755639 0.75 CYP1A2 (0.48) ALDH1A1POLBTDP1L3MBTL1MEN1
SCHEMBL5758300 0.73 ALDH1A1 (0.50) ALDH1A1KMT2AKDM4EMAPTLMNA
SCHEMBL20697505 0.72 TSHR (0.47) ALDH1A1POLBTDP1L3MBTL1APEX1
SCHEMBL17059031 0.71 HSD17B10 (0.49) ALDH1A1HSD17B10MEN1KMT2AMPI

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009136663-A1 FUSED HETEROCYCLIC DERIVATIVES AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-11-12 WO disclosed