SCHEMBL5761749

SCHEMBL5761749

CN(C(=O)C1CCN(C(=O)O)C(Cc2ccccc2)C1)C(c1ccnc(F)c1)C(O)c1cccc(C(F)(F)F)c1

nearest known ligand 0.38

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 11/20 0.38
OPRK1 P41145 1/20 0.37
GRIN2B Q13224 1/20 0.36
CETP P11597 5/20 0.35
CHRM4 P08173 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5761752 0.82 SMN1; SMN2 (0.42) TACR1OPRK1GRIN2BCHRM4
SCHEMBL6280979 0.70 GRIN2B (0.42) GRIN2B
SCHEMBL3075266 0.70 TACR1 (0.50) TACR1
SCHEMBL7994460 0.70 FOLH1 (0.37) OPRK1
SCHEMBL5201104 0.70 EPHX1 (0.40) CHRM4
SCHEMBL2199235 0.66 TACR1 (0.41) TACR1
SCHEMBL581462 0.64 NOTUM (0.49) TACR1
SCHEMBL6952343 0.64 L3MBTL1 (0.49) TACR1
SCHEMBL581110 0.63 TACR1 (0.48) TACR1
SCHEMBL206989 0.63 TACR1 (0.46) TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1414443-B1 BENZIMIDAZO 4,5-f|ISOQUINOLINONE DERIVATIVES MERCK & CO INC (US) 2006-11-15 EP disclosed