SCHEMBL5762893

SCHEMBL5762893

N#C[C@]1(c2ccccc2NC(=O)OCc2ccccc2)C2CCC[C@@H]21

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.49
RAB9A P51151 1/20 0.49
PREP P48147 4/20 0.45
CASP3 P42574 1/20 0.44
CTSL P07711 3/20 0.43
CTSB P07858 3/20 0.43
CTSK P43235 2/20 0.43
ALDH1A1 P00352 2/20 0.43
CTSS P25774 2/20 0.42
GAA P10253 1/20 0.41
MAOB P27338 3/20 0.41
KDM1A O60341 2/20 0.41
MAOA P21397 2/20 0.41
POLB P06746 1/20 0.41
MMP2 P08253 2/20 0.40
MMP9 P14780 2/20 0.40
RCOR1 Q9UKL0 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5764459 0.82 KDM1A (0.51) NPC1RAB9APREPCTSLCTSB
SCHEMBL6002580 0.82 KDM1A (0.51) NPC1RAB9APREPCTSLCTSB
SCHEMBL5764315 0.80 NPC1 (0.43) NPC1RAB9APREPCASP3CTSL
SCHEMBL541864 0.70 ALDH1A1 (0.58) NPC1RAB9ACASP3ALDH1A1GAA
SCHEMBL2233522 0.68 NPC1 (0.69) NPC1RAB9ACASP3ALDH1A1MAOB
SCHEMBL16193532 0.68 NPC1 (0.69) NPC1RAB9ACASP3MAOBPOLB
SCHEMBL30522295 0.68 NPC1 (0.69) NPC1RAB9ACASP3MAOBPOLB
SCHEMBL29950689 0.68 NPC1 (0.64) NPC1RAB9ACASP3ALDH1A1MAOB
SCHEMBL4291027 0.68 NPC1 (0.64) NPC1RAB9ACASP3ALDH1A1MAOB
SCHEMBL7982809 0.67 NPC1 (0.50) NPC1RAB9ACASP3KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1656357-A1 OXAZOLIDINONE ANTIBIOTICS AND DERIVATIVES THEREOF Merck & Co., Inc. (US) 2006-05-17 EP disclosed
WO-2005005399-A1 OXAZOLIDINONE ANTIBIOTICS AND DERIVATIVES THEREOF MERCK & CO., INC. (US) 2005-01-20 WO disclosed