SCHEMBL5763201

SCHEMBL5763201

O=C1COc2ccc(C(O)CN3CCC(C(=O)O)CC3)cc2N1

nearest known ligand 0.48

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.48
TRPV1 Q8NER1 12/20 0.47
DRD2 P14416 2/20 0.44
DRD4 P21917 2/20 0.44
GAA P10253 1/20 0.43
ALDH1A1 P00352 1/20 0.43
MAPT P10636 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5655518 1.00 PARP1 (0.48) PARP1TRPV1DRD2DRD4GAA
SCHEMBL5774775 0.85 DRD4 (0.46) PARP1DRD2DRD4GAAALDH1A1
SCHEMBL3783255 0.84 PARP1 (0.45) PARP1DRD2DRD4ALDH1A1MAPT
SCHEMBL5657579 0.79 HTT (0.46) TRPV1DRD2ALDH1A1MAPT
SCHEMBL5659963 0.79 AOC3 (0.46) ALDH1A1
SCHEMBL5659968 0.79 AOC3 (0.46) ALDH1A1
SCHEMBL5659998 0.79 ALDH1A1 (0.59) PARP1TRPV1GAAALDH1A1MAPT
SCHEMBL5658401 0.79 HTR1A (0.58) PARP1DRD2DRD4
SCHEMBL3786601 0.77 ALDH1A1 (0.47) PARP1DRD2DRD4GAAALDH1A1
SCHEMBL4759018 0.76 DRD2 (0.44) PARP1DRD2DRD4GAAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1392686-B1 BICYCLIC NITROGEN-CONTAINING HETEROCYCLIC DERIVATIVES FOR USE AS ANTIBACTERIALS SMITHKLINE BEECHAM PLC (GB) 2006-10-18 EP disclosed